An antifungal agent is a drug that selectively eliminates fungal pathogens from a host with minimal toxicity to the host. Classes: 1. Polyene Antifungal Drugs: Amphotericin, nystatin, and pimaricin interact with sterols in the cell membrane (ergosterol in fungi, cholesterol in humans) to form channels through which small molecules leak from the inside of the fungal cell to the outside. 2. Azole Antifungal Drugs: Fluconazole, itraconazole, and ketoconazole inhibit cytochrome P450-dependent enzymes (particularly C14-demethylase) involved in the biosynthesis of ergosterol, which is required for fungal cell membrane structure and function. 3. Allylamine and Morpholine Antifungal Drugs: lylamines (naftifine, terbinafine) inhibit ergosterol biosynthesis at the level of squalene epoxidase. The morpholine drug, amorolfine, inhibits the same pathway at a later step. 4. Antimetabolite Antifungal Drugs: 5-Fluorocytosine acts as an inhibitor of both DNA and RNA synthesis via the intracytoplasmic conversion of 5-fluorocytosine to 5-fluorouracil.


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4'-Hydroxy-2,4-dimethoxychalcone

4'-Hydroxy-2,4-dimethoxychalcone is a natural chalcone derivatives in the red herbal resin of Dracaena cochinchinensis. 4'-Hydroxy-2,4-dimethoxychalcone displays a wide range of biological activities including antimalarial, antiprotozoal, antibacterial, antifungal activity[1][2].

  • CAS Number: 151135-64-7
  • MF: C17H16O4
  • MW: 284.306
  • Catalog: Bacterial
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 500.1±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 185.8±23.6 °C

S-F24

S-F24 is an antifungal agent with excellent broad-spectrum. S-F24 inhibits CYP3A4 with an IC50 value of 0.4 μM. S-F24 displays a good safety profile with high selectivity, low hemolytic effects, and low tendency to induce resistance. S-F24 can be used for research on fungal infections[1].

  • CAS Number: 2946669-78-7
  • MF: C25H27BrF2N6O
  • MW: 545.42
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Picropodopyllotoxone

Picropodophyllone, an aryltetralin lignan, is isolated from leaves of Podophyllum hexandrum, and has antifungal activities[1][2].

  • CAS Number: 477-48-5
  • MF: C22H20O8
  • MW: 412.38900
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: 602.3±55.0 °C at 760 mmHg
  • Melting Point: 153-154 °C
  • Flash Point: N/A

(2α,3α)-2,3,24-Trihydroxyurs-12-en-28-oic acid

Pygenic acid B is a triterpenoid that can be isolated from the leaves of Glochidion obliquum. Pygenic acid B shows antifungal activity against C. musae. Pygenic acid B shows ONOO- scavenging activity[1][2][3].

  • CAS Number: 89786-83-4
  • MF: C30H48O5
  • MW: 488.699
  • Catalog: Fungal
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 609.4±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 336.4±28.0 °C

Eberconazole

Eberconazole is a dichlorinated imidazole derivative with antifungal activity. Eberconazole is more active than Clotrimazole, Ketoconazole, and Miconazole. Eberconazole has the potential for the research of dermatophytoses with a topical administration[1].

  • CAS Number: 128326-82-9
  • MF: C18H14Cl2N2
  • MW: 329.22300
  • Catalog: Fungal
  • Density: 1.35g/cm3
  • Boiling Point: 495ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 253.2ºC

Seselin

Seselin is an anticancer, antinociceptive, anti-inflammatory and antifungal agent. Seselin is orally active[1][2][3].

  • CAS Number: 523-59-1
  • MF: C14H12O3
  • MW: 228.24
  • Catalog: Fungal
  • Density: 1.222g/cm3
  • Boiling Point: 403ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 170.5ºC

Antibacterial agent 73

Antibacterial agent 73 (compound 7a) is a potent antimicrobial agent. Antibacterial agent 73 exhibits very good antitubercular activity (MIC=0.65 µg/mL) against Mtb H37Rv. Antibacterial agent 73 shows good activity against fungal and bacterial. Antibacterial agent 73 also shows cytotoxicity in MCF-7 breast cancer cell lines, with IC50 of 8.20 μM[1].

  • CAS Number: 414885-92-0
  • MF: C15H17FN2O
  • MW: 260.31
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-Methoxyberberium

1-Methoxyberberine chloride is a plant alkaloid that can be found in Corydalis longipes. 1-Methoxyberberine chloride exhibits antifungal effects[1].

  • CAS Number: 29133-52-6
  • MF: C21H20ClNO5
  • MW: 401.84
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Chlormidazole hydrochloride

Chlormidazole hydrochloride is an antifungal agent and has inhibitory activity against many fungi and some gram-positive cocci. Chlormidazole hydrochloride can be applied in fungal and bacterial infections of nails and skin, including interdigital and periungual mycoses[1].

  • CAS Number: 74298-63-8
  • MF: C15H14Cl2N2
  • MW: 293.19100
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: 467.5ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 236.5ºC

Dehydroacetic acid sodium

Dehydroacetic acid sodium, a pyrone derivative acts as an antibacterial and antifungal agent. Dehydroacetic acid possess phytotoxic activity[1].

  • CAS Number: 4418-26-2
  • MF: C8H7NaO4
  • MW: 190.128
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: 332.6ºC at 760 mmHg
  • Melting Point: ~295 °C (dec.)
  • Flash Point: 150.6ºC

5-hydroxymethylfurfural

5-(Hydroxymethyl)furan-2-carbaldehyde, derived from lignocellulosic biomass, inhibits yeast growth and fermentation as stressors.

  • CAS Number: 67-47-0
  • MF: C6H6O3
  • MW: 126.110
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 291.5±30.0 °C at 760 mmHg
  • Melting Point: 28-34 °C(lit.)
  • Flash Point: 79.4±0.0 °C

PD 113270

PD 113270 (CL 1565-B) is an antitumor agent. PD 113270 exhibits inhibitory effects to yeasts[1].

  • CAS Number: 87860-37-5
  • MF: C19H27O8P
  • MW: 414.38700
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Lawsone methyl ether

Lawsone methyl ether (2-Methoxy-1,4-naphthoquinone), isolated from Impatiens balsamina L. and Swertia calycina, exhibits potent antifungal and antibacterial activities[1].

  • CAS Number: 2348-82-5
  • MF: C11H8O3
  • MW: 188.17900
  • Catalog: Bacterial
  • Density: 1.28g/cm3
  • Boiling Point: 339.8ºC at 760mmHg
  • Melting Point: 184-187ºC(lit.)
  • Flash Point: 152.7ºC

Aurachin D

Aurachin D is an antibiotic. Aurachin D inhibits Gram-positive bacteria and a few funguses. Aurachin D blocks NADH oxidation in beef heart submitochondrial particles[1].

  • CAS Number: 108354-13-8
  • MF: C25H33NO
  • MW: 363.54
  • Catalog: Bacterial
  • Density: 0.981g/cm3
  • Boiling Point: 492.3ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 130.2ºC

Swinholide A

Swinholide A is the actin-binding marine polyketide and dimerizes actin with the Kd of ~ 50 nM[1]. Swinholide A is a microfilament disrupting marine toxin that stabilizes actin dimers and severs actin filaments. Swinholide A disrupts the actin cytoskeleton of cells.Antifungal activity[2].

  • CAS Number: 95927-67-6
  • MF: C78H132O20
  • MW: 1389.87
  • Catalog: Fungal
  • Density: 1.15 g/cm3
  • Boiling Point: 1249.8ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 307.3ºC

N-(4-Bromo-2-methyl-phenyl)-2-chloro-acetamide

2-Chloro-N-(2-methyl-4-bromophenyl)acetamide is an antifungal compound[1].

  • CAS Number: 96686-51-0
  • MF: C9H9BrClNO
  • MW: 262.53
  • Catalog: Fungal
  • Density: 1.578g/cm3
  • Boiling Point: 372.3ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 179ºC

Enfumafungin

Enfumafungin, a triterpene glycoside, is isolated from extracts derived from an endophytic species of Hormonema. Enfumafungin is an antifungal compound that is acting on the fungal cell wall, as the (1,3)-beta-D-glucan synthase inhibitor. Enfumafungin is specific for yeasts and fungi (excluding Cryptococcus) and does not inhibit the growth of Bacillus subtilis[1][2].

  • CAS Number: 260979-95-1
  • MF: C38H60O12
  • MW: 708.88
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Neophellamuretin

Neophellamuretin is a flavonoid. Neophellamuretin inhibits Trichophyton sp. with an MIC value of 62.5 µg/mL[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Dermaseptin

Dermaseptin-S1 is an antimicrobial peptide derived from frog skin against filamentous fungi[1].

  • CAS Number: 136033-70-0
  • MF: C152H257N43O44S2
  • MW: 3455.059
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 2954.0±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 1740.3±34.3 °C

Antifungal agent 77

Antifungal agent 77 (Compound 13h) is an antifungal agent. Antifungal agent 77 (500 μg/mL) also shows good insecticidal activity against Mythimna separate, Helicoverpa armigera, Ostrinia nubilalis, and Spodoptera frugiperda with a death rate of 30%, 25%, 40%, and 25%. Antifungal agent 77 shows toxicity in zebrafish embryo with a LC50 of 2.43 μg/mL[1].

  • CAS Number: 2863678-89-9
  • MF: C21H18FN5O2
  • MW: 391.40
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Inz-5

Inz-5 is a fungal-selective mitochondrial cytochrome bc1 inhibitor. Inz-5 impairs fungal virulence and prevents the evolution of drug resistance[1].

  • CAS Number: 1585214-21-6
  • MF: C18H14F4N6
  • MW: 390.34
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Rhamnolipid RL2

Rhamnolipid RL2, is a rhamnolipid, shows antifungal activity[1][2].

  • CAS Number: 4348-76-9
  • MF: C32H58O13
  • MW: 650.79500
  • Catalog: Fungal
  • Density: 1.23g/cm3
  • Boiling Point: 798.8ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 243.4ºC

Caerulomycin A

Caerulomycin A (Cerulomycin; Caerulomycin), an antifungal compound, induces generation of T cells, enhances TGF-β-Smad3 protein signaling via suppressing interferon-γ-induced STAT1 signaling. Antifungal and antibiotic activity, and used in autoimmune diseases[1].

  • CAS Number: 21802-37-9
  • MF: C12H11N3O2
  • MW: 229.23500
  • Catalog: Fungal
  • Density: 1.23g/cm3
  • Boiling Point: 400.4ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 195.9ºC

kievitone

Kievitone, an isoflavanone, could be isolated from hypocotyls of Phaseolus vulgaris L. infected with Rhizoctonia solani Kühn. Kievitone has antifungal activity and antitumor activity[1][2].

  • CAS Number: 40105-60-0
  • MF: C20H20O6
  • MW: 356.36900
  • Catalog: Fungal
  • Density: 1.384g/cm3
  • Boiling Point: 639.6ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 231.4ºC

Aloin

Aloin (mixture of A&B) is anthraquinone derivative isolated from Aloe vera. Aloin (mixture of A&B) has diverse biological activities such as anti-inflammatory, immunity, antidiabetic, antioxidant, antibacterial, antifungal, and antitumor activities. Aloin (mixture of A&B) also an effective inhibitor of stimulated granulocyte matrix metalloproteinases (MMPs)[1][2].

  • CAS Number: 8015-61-0
  • MF: C21H22O9
  • MW: 418.394
  • Catalog: Bacterial
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: 752.6±60.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 268.0±26.4 °C

Isoprothiolane-d4

Isoprothiolane-d4 is the deuterium labeled Isoprothiolane. Isoprothiolane is a systemic fungicide. Isoprothiolane is a rice blast controlling agent against the fungal disease of rice planty Pyvioutavia oryzae Cav[1][2].

  • CAS Number: 1715020-82-8
  • MF: C12H14D4O4S2
  • MW: 294.42
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Metalaxyl-M

Metalaxyl-M ((R)-Metalaxyl) is the active (R)-enantiomer of Metalaxyl. Metalaxyl-M is a broad-spectrum fungicide that inhibits protein and ribosomal RNA synthesis in fungi. Metalaxyl is used for research of plant diseases caused by pathogens of the Oomycota division[1].

  • CAS Number: 70630-17-0
  • MF: C15H21NO4
  • MW: 279.33200
  • Catalog: Fungal
  • Density: 1.117 g/cm3
  • Boiling Point: 394.3ºC at 760 mmHg
  • Melting Point: 38.7ºC
  • Flash Point: 192.3ºC

Antifungal agent 32

Antifungal agent 32 (compound 1a) is a potent antifungal agent. Antifungal agent 32 inhibits Candida albicans filamentation and biofilm formation. Antifungal agent 32 inhibits the morphological switching of Candida albicans and its adherence to epithelial cells. Antifungal agent 32 can be used for Candida albicans infections research[1].

  • CAS Number: 1809167-48-3
  • MF: C25H28N2O
  • MW: 372.50
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

4-Isopropylbenzoic acid

4-Isopropylbenzoic acid, an aromatic monoterpenoid, is isolated from the stem bark of Bridelia retusa. 4-Isopropylbenzoic acid exhibits antifungal activities. 4-Isopropylbenzoic acid is also a reversible and uncompetitive inhibitor of mushroom tyrosinase[1][2].

  • CAS Number: 536-66-3
  • MF: C10H12O2
  • MW: 164.201
  • Catalog: Fungal
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 271.8±19.0 °C at 760 mmHg
  • Melting Point: 117-120 °C(lit.)
  • Flash Point: 128.1±16.2 °C

Acetyleugenol

Eugenol acetate (Eugenyl acetate), a major phytochemical constituent of the essential oil exhibits antibacterial, antioxidant, and anti-virulence activities. Eugenol acetate (Eugenyl acetate), a phytochemical in clove essential oil, against clinical isolates of Candida albicans, Candida parapsilosis, Candida tropicalis, and Candida glabrata.

  • CAS Number: 93-28-7
  • MF: C12H14O3
  • MW: 206.238
  • Catalog: Bacterial
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 268.0±28.0 °C at 760 mmHg
  • Melting Point: 26°C
  • Flash Point: 106.8±18.6 °C