Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

MEL24

MEL24 is an Mdm2 E3 ligase inhibitor that reduces cell survival and increases sensitivity to DNA damaging agents in a p53-dependent manner for in vitro antitumor studies[1].

  • CAS Number: 642072-48-8
  • MF: C17H18N4O3
  • MW: 326.35
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Peptide ε

Protein Kinase C Peptide Substrate is targeted to a specific cellular compartment in a manner dependent on second messengers and on specific adapter proteins in response to extracellular signals that activate G-protein-coupled receptors, tyrosine kinase receptors, or tyrosine kinase-coupled receptors. Protein Kinase C Peptide Substrate then regulates various physiological functions including the activation of nervous, endocrine, exocrine, inflammatory, and immune systems[1].

  • CAS Number: 120253-69-2
  • MF: C83H155N39O21S
  • MW: 2067.43
  • Catalog: Endocrinology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

NQTrp

NQTrp, an aromatic naphthoquinone-tryptophan hybrid molecule, an inhibitor of the aggregation of the tau protein with generic anti-amyloidogenic effects. NQTrp inhibits the in vitro aggregation of hexapeptide (41GCWMLY46 within the N-terminus of γD-crystallin) as well as full-length γD-crystallin[1].

  • CAS Number: 185351-19-3
  • MF: C21H16N2O4
  • MW: 360.36300
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Anemarrhenasaponin A2

Anemarrhenasaponin A2 (Schidigerasaponin F2;Timosaponin AII) is a steroidal saponin isolated from the rhizomes of Anemarrhena asphodeloides. Anemarrhenasaponin A2 inhibits ADP-induced platelet aggregation[1].

  • CAS Number: 117210-12-5
  • MF: C39H64O14
  • MW: 756.92
  • Catalog: Cardiovascular Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Acetamide,N,N-diphenyl-

N,N-Diphenylacetamide (N-Acetyldiphenylamine) has N,N-disubstituted amide group and can be used as a mono- as well as a bidentate ligand generating four-membered chelate rings[1].

  • CAS Number: 519-87-9
  • MF: C14H13NO
  • MW: 211.26
  • Catalog: Others
  • Density: 1.125g/cm3
  • Boiling Point: 130 °C0.02 mm Hg(lit.)
  • Melting Point: 100-103 °C(lit.)
  • Flash Point: 199.7ºC

Ruzadolane

Ruzadolane is a non-narcotic, centrally-acting analgesic agent.

  • CAS Number: 115762-17-9
  • MF: C18H19F2N5S
  • MW: 375.43900
  • Catalog: Neurological Disease
  • Density: 1.38g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

iNOs-IN-3

iNOs-IN-3 (Compound 2d) is an orally active nitric oxide synthase (iNOS) inhibitor (IC50=3.342 µM). iNOs-IN-3 shows anti-inflammatory activity and can be used in LPS-induced acute lung injury (ALI) research[1].

  • CAS Number: 2241674-94-0
  • MF: C27H24N2O5S
  • MW: 488.55
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-Lys(Biotin)-OH

Fmoc-Lys(Biotin)-OH is a lysine derivative[1].

  • CAS Number: 146987-10-2
  • MF: C31H38N4O6S
  • MW: 594.722
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 936.2±65.0 °C at 760 mmHg
  • Melting Point: 183 °C
  • Flash Point: 520.0±34.3 °C

cepharanoline

Cepharanoline is a compound isolated from Stephania cepharantha Hayata. Cepharanoline has proliferative activities[1].

  • CAS Number: 27686-34-6
  • MF: C36H36N2O6
  • MW: 592.68100
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

3-Cyclopentyl-DL-alanine

3-DL-Cpa-OH is an alanine derivative[1].

  • CAS Number: 96539-87-6
  • MF: C8H15NO2
  • MW: 157.210
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 290.5±23.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 129.5±22.6 °C

Chlorempenthrin

Chlorempenthrin is a synthetic pyrethroid insecticide[1].

  • CAS Number: 54407-47-5
  • MF: C17H22Cl2O2
  • MW: 329.261
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 399.5±42.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 136.8±26.9 °C

(1Z,5Z,9Z)-14-benzyl-12-hydroxy-4,6,15,15a-tetramethyl-8,11-dioxo-4,7,8,11,14,14a,15,15a,16a,16b-decahydro-3H-cyclotrideca[d]oxireno[2,3-f]isoindol-7-yl acetate

Cytochalasin K (Compounds 7) is a cytochalasin that inhibits wheat root elongation with an IC50 of 22.58 μM[1].

  • CAS Number: 79648-72-9
  • MF: C32H37NO6
  • MW: 531.63900
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

N-Acetyl-S-[3-acetamino-6-hydroxphenyl]-cysteine allyl ester-d5

N-Acetyl-S-[3-acetamino-6-hydroxphenyl]-cysteine allyl ester-d5 is the deuterium labeled N-Acetyl-S-[3-acetamino-6-hydroxphenyl]-cysteine allyl ester[1].

  • CAS Number: 1331889-45-2
  • MF: C16H15D5N2O5S
  • MW: 357.44
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

MAT2A inhibitor 3

MAT2A inhibitor 3 is a methionine adenosyltransferase 2A (MAT2A) inhibitor extracted from patent WO2020123395A1, compound 24, has an IC50 of <200 nM. MAT2A inhibitor 3 can be used for the research of cancers[1].

  • CAS Number: 2439271-82-4
  • MF: C16H14ClN3O
  • MW: 299.75
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1,3,5-Tribromobenzene-d3

1,3,5-Tribromobenzene-d3 is the deuterium labeled 1,3,5-Tribromobenzene[1].

  • CAS Number: 52921-77-4
  • MF: C6Br3D3
  • MW: 317.81900
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

L-Rhamnose

α-L-Rhamnose monohydrate is a component of the plant cell wall pectic polysaccharides rhamnogalacturonan I and rhamnogalacturonan II. α-L-Rhamnose monohydrate is also a component of bacterial polysaccharides where it plays an important role in pathogenicity.

  • CAS Number: 6155-35-7
  • MF: C6H14O6
  • MW: 182.172
  • Catalog: Infection
  • Density: N/A
  • Boiling Point: 323.9ºC at 760 mmHg
  • Melting Point: 90-95ºC
  • Flash Point: 149.7ºC

Triphenylamine-d15

Triphenylamine-d15 is the deuterium labeled Triphenylamine[1].

  • CAS Number: 880462-20-4
  • MF: C18H15N
  • MW: 245.31800
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Methyl (3α)-3,27-dihydroxylup-20(29)-en-28-oate

Antiproliferative agent-29 (Compound 16) is a triterpenoid isolated from the seeds of Peganum harmala L. Antiproliferative agent-29 has antiproliferative activity and has potential for cancer research[1].

  • CAS Number: 263844-79-7
  • MF: C31H50O4
  • MW: 486.73
  • Catalog: Cancer
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 557.1±25.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 169.3±16.7 °C

Amyloid β-Protein (1-24) trifluoroacetate salt

Amyloid β-Protein (1-24) is a biologically active peptide.

  • CAS Number: 138648-77-8
  • MF: C130H183N35O40
  • MW: 2876.054
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Caulophyllumine A

Caulophyllumine A is a natural product that can be isolated from blue cohosh[1].

  • CAS Number: 1009318-60-8
  • MF: C15H21NO4
  • MW: 279.332
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 451.8±40.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 227.0±27.3 °C

Efprezimod alfa

Efprezimod alfa is an active peptide. Efprezimod alfa can be used for various biochemical studies.

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

HC-056456

HC-056456 is an effective but not perfectly-selective blocker of CatSper channels. The [Na+]i rise is slowed by HC-056456 (IC50~3 µM).

  • CAS Number: 7733-96-2
  • MF: C12H6N2O4S2
  • MW: 306.31700
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Rocaglaol

Rocaglaol induces apoptosis and cell cycle arrest in LNCaP cells[1].

  • CAS Number: 147059-46-9
  • MF: C26H26O6
  • MW: 434.48
  • Catalog: Cancer
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 584.6±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 307.3±30.1 °C

Monochlorobimane

Monochlorobimane is a fluorescent dye (λex=380 nm, λem=470 nm).

  • CAS Number: 76421-73-3
  • MF: C10H11ClN2O2
  • MW: 226.66000
  • Catalog: Dye Reagents
  • Density: 1.4g/cm3
  • Boiling Point: 314.9ºC at 760 mmHg
  • Melting Point: 135-136ºC(lit.)
  • Flash Point: 144.2ºC

Cistanoside F

Cistanoside F is a phenylethanoid glycosid isolated from Cistanche deserticola, with antioxidative effect[1].

  • CAS Number: 97411-47-7
  • MF: C21H28O13
  • MW: 488.439
  • Catalog: Others
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: 880.7±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 302.8±27.8 °C

Dielaidoylphosphatidylethanolamine

Dielaidoylphosphatidylethanolamine is a liposome used to deliver drugs[1].

  • CAS Number: 16777-83-6
  • MF: C41H78NO8P
  • MW: 744.03400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Scopoline

Scopoline (compound 3a) is a compound easily formed from scopine[1].

  • CAS Number: 487-27-4
  • MF: C8H13NO2
  • MW: 155.19
  • Catalog: Others
  • Density: 1.284 g/cm3
  • Boiling Point: 248ºCat 760 mmHg
  • Melting Point: 107-109ºC
  • Flash Point: 111.6ºC

Dap-NE hydrochloride (GMP)

Dap-NE hydrochloride (GMP) is Dap-NE hydrochloride (HY-78932A) produced by using GMP guidelines. Dap-NE hydrochloride is an intermediate used in the synthesis of antibody-drug conjugates (ADCs)[1].

  • CAS Number: 2019182-02-4
  • MF: C18H29ClN2O3
  • MW: 356.88746
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Oleuroside

Oleuroside is a phenolic secoiridoid in olive. Oleuroside can protect against mitochondrial dysfunction in models of early Alzheimer's disease and brain ageing[1].

  • CAS Number: 116383-31-4
  • MF: C25H32O13
  • MW: 540.52
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

H-Gly-Ser-OH

Glycyl-l-serine is a serine derivative[1].

  • CAS Number: 7361-43-5
  • MF: C5H10N2O4
  • MW: 162.144
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 513.0±50.0 °C at 760 mmHg
  • Melting Point: 201-202℃
  • Flash Point: 264.1±30.1 °C