Opioid receptors are a group of G protein-coupled receptors with opioids as ligands. The endogenous opioids are dynorphins, enkephalins, endorphins, endomorphins and nociceptin. Opioid receptors are distributed widely in the brain, and are found in the spinal cord and digestive tract. Opioid receptors are molecules, or sites, within the body that are activated by opioid substances. Opioid receptors inhibit the transmission of impulse in excitatory pathways within the human body system. These pathways include the serotonin, catecholamine, and substance P pathways, which are all implicated in pain perception and feelings of well-being. Opioid receptors are further subclassified into mu, delta, and kappa receptors. All the classes, while exhibiting differing modes of action, share some basic similarities. They all are driven by the potassium pump mechanism, which is found on the plasma membrane of the majority of cells.


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β-Casomorphin, bovine

β-casomorphin, bovine (β-casomorphin-7) is a opioid peptide with an IC50 of 14 μM in an Opioid receptors binding assay.

  • CAS Number: 72122-62-4
  • MF: C41H55N7O9
  • MW: 789.91700
  • Catalog: Peptides
  • Density: 1.32g/cm3
  • Boiling Point: 1170.5ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 661.7ºC

(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) trifluoroacetate salt

(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) (E-2078), a stable Dynorphin A (1–8) (HY-P2159) analog, is a kappa opioid receptor (KOR) agonist[1].

  • CAS Number: 103613-84-9
  • MF: C50H81N15O9
  • MW: 1036.273
  • Catalog: Opioid Receptor
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

BAM-22P

BAM-22P, a highly potent opioid peptide, is a potent opioid agonist.

  • CAS Number: 76622-26-9
  • MF: C130H184N38O31S2
  • MW: 2839.22000
  • Catalog: Peptides
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

ML 190

ML 190 is a selective κ opioid receptor (KOR) antagonist with an IC50 of 120 nM and an EC50 of 129 nM, respectively[1].

  • CAS Number: 1355244-02-8
  • MF: C27H32N6O3
  • MW: 488.58
  • Catalog: Opioid Receptor
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

ICI 204,448 hydrochloride

ICI-204448 is a κ-opioid agonist with limited access to the CNS, ICI-204448 can displace the binding of the kappa-opioid ligand 3H-bremazocine from guinea pig cerebellum membranes[1].

  • CAS Number: 121264-04-8
  • MF: C23H27Cl3N2O4
  • MW: 501.83
  • Catalog: Opioid Receptor
  • Density: N/A
  • Boiling Point: 638.9ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 340.2ºC

D-Ala-Gly-Phe-Met-NH2

D-Ala-Gly-Phe-Met-NH2, an opioid peptide, is a potent opiate δ-receptor agonist[1].

  • CAS Number: 82948-89-8
  • MF: C19H29N5O4S
  • MW: 423.53
  • Catalog: Opioid Receptor
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

[Arg14,Lys15] Nociceptin

[Arg14,Lys15]Nociceptin is a highly potent and selective NOP receptor agonist, with an EC50 of 1 nM. [Arg14,Lys15]Nociceptin displays high selectivity over opioid receptors, with IC50s of 0.32, 280, >10000 and 1500 nM for NOP (ORL1; OP4), μ, δ and κ receptors, respectively[1].

  • CAS Number: 236098-40-1
  • MF: C82H137N31O22
  • MW: 1909.16000
  • Catalog: Opioid Receptor
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

DPI-3290

DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively。DPI-3290 is one of a series of novel centrally acting agents with potent antinociceptive activity[1].

  • CAS Number: 182417-73-8
  • MF: C30H34FN3O2
  • MW: 487.60800
  • Catalog: Opioid Receptor
  • Density: 1.161±0.06 g/cm3(Predicted)
  • Boiling Point: 620.4±55.0 °C(Predicted)
  • Melting Point: 144-145 °C
  • Flash Point: N/A

Nociceptin(Orphanin FQ)

Nociceptin, a heptadecapeptide, is the endogenous ligand of the nociceptin receptor, acting as a potent anti-analgesic.

  • CAS Number: 170713-75-4
  • MF: C79H129N27O22
  • MW: 1809.037
  • Catalog: Peptides
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(D-Ala2)-Leu-Enkephalin

[D-Ala2]leucine-enkephalin, a delta opioid agonist, is a degradation resistant long-acting Leu-enkephalin. Sequence: Tyr-D-Ala-Gly-Phe-Leu.

  • CAS Number: 64963-01-5
  • MF: C29H39N5O7
  • MW: 569.649
  • Catalog: Peptides
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 991.9±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 553.7±34.3 °C

picraline

Picraline is a natural alkaloid that targets opioid receptors with binding affinities with Ki values of 132 μM, 2.38 μM and 98.8 μM for μOR, κOR and δOR, respectively[1].

  • CAS Number: 2671-32-1
  • MF: C23H26N2O5
  • MW: 410.46
  • Catalog: Opioid Receptor
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 548.0±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 285.2±30.1 °C

σ1 Receptor/μ Opioid receptor modulator 1

σ1 Receptor/μ Opioid receptor modulator 1 (Compound 44) is a potent σ1 receptor antagonist and μ opioid receptor agonist with Kis of 1.86 nM and 2.1 nM, respectively.σ1 Receptor/μ Opioid receptor modulator 1 exhibits potent analgesic activity. σ1 Receptor/μ Opioid receptor modulator 1 can be used for the research of neuropathic pain[1].

  • CAS Number: 2412700-00-4
  • MF: C24H31FN2O2
  • MW: 398.51
  • Catalog: Opioid Receptor
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A