Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Insulin-Like Growth Factor I (30-41)

IGF-I (30-41) is amino acids 30 to 41 fragment of Insulin-like Growth Factor I (IGF-I). IGF-I is partly responsible for systemic GH activities although it possesses a wide number of own properties (anabolic, antioxidant, anti-inflammatory and cytoprotective actions)[1].

  • CAS Number: 82177-09-1
  • MF: C51H83N19O19
  • MW: 1266.34
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

SPH5030

SPH5030 is a selective, potent, and irreversible HER2 mutants inhibitor with IC50 of <1 nM against HER2 D769H, D769Y, V777L and R896C mutants.SPH5030 exhibits high relative HER2 selectivity compared with neratinib and pyrotinib.SPH5030 shows significant in vivo antitumor efficacy in xenograft mouse models, especially in a HER2 mutation A775_G776insYVMA xenograft mouse mode.

  • CAS Number: 2364326-23-6
  • MF: C31H31FN8O3
  • MW: 582.61
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

6-FAM-PEG3-Azide

6-FAM-PEG3-Azide is a fluorescent dye that can be used to label oligonucleotide[1].

  • CAS Number: 412319-45-0
  • MF: C29H28N4O9
  • MW: 576.56
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

H-Phg-OH

H-Phg-OH is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 2935-35-5
  • MF: C8H9NO2
  • MW: 151.163
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 288.7±28.0 °C at 760 mmHg
  • Melting Point: >300 °C(lit.)
  • Flash Point: 128.4±24.0 °C

Rocuronium

Rocuronium (Org-9426) is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia.

  • CAS Number: 143558-00-3
  • MF: C32H53N2O4
  • MW: 529.77
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Angelic acid

Angelic Acid is a substance found in the essential oil of Anthemis nobilis, and it exists in an ester form. Angelic acid aids in wound healing and exhibits sedative and psychotropic properties[1].

  • CAS Number: 565-63-9
  • MF: C5H8O2
  • MW: 100.116
  • Catalog: Neurological Disease
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 198.5±0.0 °C at 760 mmHg
  • Melting Point: 44ºC
  • Flash Point: 95.9±9.6 °C

Chlorpheniramine

Chlorpheniramine is a H1 antihistamines commonly used in allergic diseases[1]. [2]. .

  • CAS Number: 132-22-9
  • MF: C16H19ClN2
  • MW: 274.78800
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 25 °C (lit.)
  • Flash Point: N/A

ONO 2506

Arundic acid (ONO-2506) is an astrocyte-modulating agent, which delays the expansion of cerebral infarcts by modulating the activation of astrocytes through inhibition of S-100β synthesis. Arundic acid (ONO-2506) has been developed as a therapeutic agent for stroke and Alzheimer’s disease[1][2][3].

  • CAS Number: 185517-21-9
  • MF: C11H22O2
  • MW: 186.29100
  • Catalog: Neurological Disease
  • Density: 0.908 g/cm3
  • Boiling Point: 289.3ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: N/A

Fumed silica

Amorphous silica can be used as an excipient, such as viscosifier, suspending agent, tablet disintegrating agent, adsorbent dispersing agent as liquid in powders. Pharmaceutical excipients, or pharmaceutical auxiliaries, refer to other chemical substances used in the pharmaceutical process other than pharmaceutical ingredients. Pharmaceutical excipients generally refer to inactive ingredients in pharmaceutical preparations, which can improve the stability, solubility and processability of pharmaceutical preparations. Pharmaceutical excipients also affect the absorption, distribution, metabolism, and elimination (ADME) processes of co-administered drugs[1].

  • CAS Number: 112945-52-5
  • MF: O2Si
  • MW: 60.08430
  • Catalog: Others
  • Density: 2.3 lb/cu.ft at 25 °C (bulk density)(lit.)
  • Boiling Point: 2230ºC
  • Melting Point: >1600°C
  • Flash Point: N/A

campestanol

Campestanol is a phytosterol that can be found in plant food. Campestanol lowers serum cholesterol and low-density lipoprotein. Campestanol can be used for the research of metabolic disorders[1].

  • CAS Number: 474-60-2
  • MF: C28H50O
  • MW: 402.70
  • Catalog: Metabolic Disease
  • Density: 0.951g/cm3
  • Boiling Point: 461.4ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 193ºC

Eicosapentaenoic Acid methyl ester

Eicosapentaenoic acid methyl ester is a degradant of a monogalactosyl diacylglycerol (an anticancer compound by inducing apoptosis)[1].

  • CAS Number: 2734-47-6
  • MF: C21H32O2
  • MW: 316.478
  • Catalog: Others
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 402.8±34.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 104.4±24.0 °C

KRN5

KRN5 is a Nuclear factor of activated T cells 5 (NFAT5) suppressor, with an IC50 of 750 nM.

  • CAS Number: 1800465-47-7
  • MF: C27H22FNO5
  • MW: 459.47
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Cimigenoside

Cimigenoside is an active compound from genus Cimicifuga[1].

  • CAS Number: 27994-11-2
  • MF: C35H56O9
  • MW: 616.782
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

GRK5-IN-2

GRK5-IN-2 (compound 707), a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor. GRK5-IN-2 regulates the expression and/or release of insulin and is useful for the metabolic disease research[1].

  • CAS Number: 1642839-27-7
  • MF: C20H20N4O4
  • MW: 380.40
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Sominone

Sominone is a withanolide. Sominone can be isolated from the herbs of Withania somnifera[1].

  • CAS Number: 98569-64-3
  • MF: C28H42O5
  • MW: 458.63000
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Zincon monosodium salt

Zincon sodium is an excellent colorimetric reagent for the detection of zinc and copper ions in aqueous solution. Zincon sodium can be used for the determination of zinc, copper, and cobalt ions in metalloproteins[1].

  • CAS Number: 62625-22-3
  • MF: C20H15N4O6S.Na
  • MW: 462.41
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: 250-260 °C (dec.)
  • Flash Point: N/A

1,4,7-Eudesmanetriol

1β,4β,7α-Trihydroxyeudesmane (compound 4) is a nature product that could be isolated from the rhizomes of Homalomena occulta. 1β,4β,7α-Trihydroxyeudesmane has antiproliferative active. 1β,4β,7α-Trihydroxyeudesmane can be used in research of cancer[1].

  • CAS Number: 145400-02-8
  • MF: C15H28O3
  • MW: 256.38
  • Catalog: Cancer
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 375.7±42.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 170.5±22.5 °C

ABL127

ABL127 is a selective and covalent inhibitor of protein methylesterase 1 (PME-1) with IC50s of 6.4 nM and 4.2 nM in HEK293T and MDA-MB-231 cells, respectively.

  • CAS Number: 1073529-41-5
  • MF: C17H20N2O5
  • MW: 332.351
  • Catalog: Cancer
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 422.8±48.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 209.5±29.6 °C
  • CAS Number: 94736-09-1
  • MF: C9H15N2NaO14P3
  • MW: 491.13100
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(Rac)-cis-3-hydroxy glyburide-13C,d3

(Rac)-cis-3-hydroxy glyburide-13C,d3 is a 13C-labeled and deuterium labeled (Rac)-cis-3-hydroxy glyburide[1].

  • CAS Number: 1217848-91-3
  • MF: C2213CH25D3ClN3O6S
  • MW: 514.01
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Tiopronin

Tiopronin is a prescription thiol drug used to control the rate of cystine precipitation and excretion in the disease cystinuria.Target: OthersTiopronin is used primarily for cystinuria and is well known in the cystinuric community. Depending on the severity of a person's cystinuria, tiopronin may be taken for life, possibly starting in early childhood. It may also be used for Wilson's disease (an overload of copper in the body), and certain types of rare arthritis, though tiopronin is not an anti-inflammatory. Tiopronin is also sometimes used as a stabilizing agent for metal nanoparticles. The thiol group binds to the nanoparticles, preventing coagulation [1, 2].

  • CAS Number: 1953-02-2
  • MF: C5H9NO3S
  • MW: 163.195
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 418.3±30.0 °C at 760 mmHg
  • Melting Point: 93-98 °C
  • Flash Point: 206.8±24.6 °C

Glycitein

Glycitein is a soybean (yellow cultivar) isoflavonoid; used in combination with other isoflavonoids such as genistein and daidzein to study apoptosis and anti-oxidation processes.

  • CAS Number: 40957-83-3
  • MF: C16H12O5
  • MW: 284.263
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 547.4±50.0 °C at 760 mmHg
  • Melting Point: >300ºC
  • Flash Point: 210.1±23.6 °C

5-Methoxy-2-benzimidazolethiol

5-Methoxy-2-benzimidazolethiol is a benzimidazole. The iodimetric determination of 5-Methoxy-2-benzimidazolethiol in alkaline media is studied[1].

  • CAS Number: 37052-78-1
  • MF: C8H8N2OS
  • MW: 180.227
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 309.4±44.0 °C at 760 mmHg
  • Melting Point: 261-263 °C(lit.)
  • Flash Point: 140.9±28.4 °C

Sodium zirconium cyclosilicate

Sodium zirconium cyclosilicate is an orally administered, non-absorbed, novel, inorganic microporous zirconium silicate compound, is a highly selective cation exchanger that selectively removes excess K+ in vivo. Sodium zirconium cyclosilicate can be used in research of chronic kidney disease (CKD)[1][2].

  • CAS Number: 17141-74-1
  • MF: H6O9Si3.2Na.Zr
  • MW: 371.50
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

D-γ-Glutamyl-D-glutamic acid

D-γ-Glutamyl-D-glutamic acid is a poly(γ-glutamic acid) of clusters of D- and D-glutamic acid repeating units in a linear chain[1].

  • CAS Number: 4553-17-7
  • MF: C10H16N2O7
  • MW: 276.24
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Ipriflavone

Ipriflavone is a synthetic isoflavone derivative used to suppress bone resorption.

  • CAS Number: 35212-22-7
  • MF: C18H16O3
  • MW: 280.318
  • Catalog: Metabolic Disease
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 435.9±45.0 °C at 760 mmHg
  • Melting Point: 116-120 °C(lit.)
  • Flash Point: 209.3±15.1 °C

H-Gly-Ala-OH

Gly-Ala is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 3695-73-6
  • MF: C5H10N2O3
  • MW: 146.145
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 417.4±30.0 °C at 760 mmHg
  • Melting Point: ~ 230°C dec.
  • Flash Point: 206.2±24.6 °C

RPRAATF

Akt/SKG Substrate Peptide is a synthetic peptide suitable as a substrate for Akt/PKB, which is not phosphorylated by p70S6K or MAPK1[1].

  • CAS Number: 276680-69-4
  • MF: C36H59N13O9
  • MW: 817.93500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

3,4,4'-Trichloro-1,1'-biphenyl-d4

3,4,4'-Trichloro-1,1'-biphenyl-d4 is the deuterium labeled 3,4,4'-Trichloro-1,1'-biphenyl[1].

  • CAS Number: 1276197-27-3
  • MF: C12H3D4Cl3
  • MW: 261.57
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

2-Methoxycinnamic acid

2-Methoxycinnamic acid is a noncompetitive inhibitor of tyrosinase[1].

  • CAS Number: 6099-03-2
  • MF: C10H10O3
  • MW: 178.185
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 325.1±17.0 °C at 760 mmHg
  • Melting Point: 182-186 °C
  • Flash Point: 130.3±14.4 °C