Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Odorinol

Odorinol is a natural product isolated from branches and leaves of Aglaia odorata. Odorinol has potential antineoplastic activity and can inhibit both the initiation and promotion stages of skin cancer[1].

  • CAS Number: 72755-22-7
  • MF: C18H24N2O3
  • MW: 316.39
  • Catalog: Cancer
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 588.6±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 309.8±30.1 °C

Atisnolerbart

Atisnolerbart is a human IgG4 antibody targeting BETVIA, the major birch pollen allergen Bet v 1-A.

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Desogestrel

Desogestrel(Org-2969) is a third-generation 19-nortestosterone derivative progestogen; is contained in many oral contraceptive preparations, both combined (COCs) to ethinyl-estradiol (EE) or alone in a progestin-only pill (POP).

  • CAS Number: 54024-22-5
  • MF: C22H30O
  • MW: 310.473
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 428.3±45.0 °C at 760 mmHg
  • Melting Point: 109-110ºC
  • Flash Point: 187.9±21.7 °C

1,5-Dichloro-2,4-dinitrobenzene-13C6

1,5-Dichloro-2,4-dinitrobenzene-13C6 is the 13C labeled 1,5-Dichloro-2,4-dinitrobenzene[1].

  • CAS Number: 335081-12-4
  • MF: C6H2Cl2N2O4
  • MW: 243.05
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

H-D-LYS(Z)-OH

H-D-Lys(Z)-OH is a lysine derivative[1].

  • CAS Number: 34404-32-5
  • MF: C14H20N2O4
  • MW: 280.320
  • Catalog: Others
  • Density: 1.206g/cm3
  • Boiling Point: 499.6±45.0 °C at 760 mmHg
  • Melting Point: 229℃
  • Flash Point: 255.9±28.7 °C

MO-I-500

MO-I-500 is a pharmacological of FTO inhibitor with an IC50 of 8.7 μM for the inhibition of purified FTO demethylase catalyzing demethylation of an artificial small methylated substrate. MO-I-500 can be used for the research of rare panresistant triple-negative inflammatory breast cancer[1].

  • CAS Number: 1585219-04-0
  • MF: C12H12ClNO5S
  • MW: 317.75
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

2-Ethylhexyl acetate-d17

2-Ethylhexyl acetate-d17 is the deuterium labeled 2-Ethylhexyl acetate[1].

  • CAS Number: 1219802-70-6
  • MF: C10H20O2
  • MW: 172.265
  • Catalog: Others
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 195.7±8.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 71.4±8.3 °C

1-Boc-4-oxo-D-proline benzyl ester

1-Boc-4-oxo-D-proline benzyl ester is a proline derivative, it can be used for the synthesis of compounds[1].

  • CAS Number: 224627-26-3
  • MF: C17H21NO5
  • MW: 319.35
  • Catalog: Others
  • Density: 1.219±0.06 g/cm3(Predicted)
  • Boiling Point: 439.9±45.0 °C(Predicted)
  • Melting Point: N/A
  • Flash Point: N/A

Ac-Pro-Leu-Gly-OH

Ac-Pro-Leu-Gly-OH is a polypeptide that can be found by peptide screening. Peptide screening is a research tool that pools active peptides primarily by immunoassay. Peptide screening can be used for protein interaction, functional analysis, epitope screening, especially in the field of agent research and development[1].

  • CAS Number: 89626-38-0
  • MF: C15H25N3O5
  • MW: 327.38
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-(azidomethyl)pyrene

1-(Azidomethyl)pyrene is a fluorescent dye[1].

  • CAS Number: 1006061-57-9
  • MF: C17H11N3
  • MW: 257.28900
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 68 °C
  • Flash Point: N/A

α-Amylase

α-Amylase from Aspergillus oryzae is an amylase. α-Amylase from Aspergillus oryzae can be used for various biochemical studies[1].

  • CAS Number: 9001-19-8
  • MF: C9H14N4O3
  • MW: 226.232
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 656.2±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 350.7±31.5 °C

DHX9-IN-3

DHX9-IN-3 (Compound 621) is an ATP-dependent inhibitor of RNA helicase A (DHX9) with potential for cancer research[1].

  • CAS Number: 2973401-57-7
  • MF: C24H20ClFN4O4S2
  • MW: 547.02
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

TMB-PS

TMB-PS(102062-36-2) is N-(3-sulfopropyl)-3,3',5,5'-tetramenthylbenzidine sodium salt; White - pale yellow crystalline powder, soluble in water, can be used under neutral, acidic and alkaline conditions.

  • CAS Number: 102062-36-2
  • MF: C19H26N2O3S
  • MW: 362.486
  • Catalog: Dye Reagents
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: 230-240ºC
  • Flash Point: N/A

Eflornithine

Eflornithine is a specific, irreversible inhibitor of the enzyme ornithine decarboxylase. Eflornithine is a medication for the treatment of African trypanosomiasis and excessive facial hair growth in women.

  • CAS Number: 70052-12-9
  • MF: C6H12F2N2O2
  • MW: 182.16800
  • Catalog: Others
  • Density: 1.293g/cm3
  • Boiling Point: 347ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 163.7ºC

AC-PHE-OET

(S)-Ethyl 2-acetamido-3-phenylpropanoate is a phenylalanine derivative[1].

  • CAS Number: 2361-96-8
  • MF: C13H17NO3
  • MW: 235.27900
  • Catalog: Others
  • Density: 1.096g/cm3
  • Boiling Point: 402.1ºC at 760mmHg
  • Melting Point: 92 °C
  • Flash Point: 197ºC

Boc-N-ethylglycine

Boc-N-Ethylglycine is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 149794-10-5
  • MF: C9H17NO4
  • MW: 203.236
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 302.7±21.0 °C at 760 mmHg
  • Melting Point: 87-88℃
  • Flash Point: 136.9±22.1 °C

Zika virus-IN-1

Zika virus-IN-1 (Compd 2) is a Zika virus inhibitor, with an EC50 of 1.56 μM [1].

  • CAS Number: 2527912-80-5
  • MF: C30H37N3O3Si
  • MW: 515.72
  • Catalog: Infection
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

IRGRILHDGAYSLTLQGLGIH

IRGRILHDGAYSLTLQGLGIH is a multi-epitope class II rat HER2/neu peptide. IRGRILHDGAYSLTLQGLGIH can be used for the research class II HER2-DC1 vaccine studies[1].

  • CAS Number: 1443436-79-0
  • MF: C102H168N32O28
  • MW: 2290.62
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

H-Pro-Pro-Pro-Pro-OH

Tetraproline is a fragment sequence in tristetraprolin (TTP). Recruitment of the 4EHP-GYF2 cap-binding complex to tetraproline motifs of tristetraprolin promotes repression and degradation of mRNAs with AU-rich elements[1].

  • CAS Number: 21866-90-0
  • MF: C20H30N4O5
  • MW: 406.48
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 729.8±60.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 395.2±32.9 °C

Cyanine 3 Tyramide

Cyanine 3 Tyramide (Tyramide-Cy3), an orange fluorescent dye, is utilized as reporter fluorescent substrate for horseradish peroxidase (HRP)-catalyzed deposition that is signal amplification technique in immunoassay and in situ hybridization of nucleic acids[1][2].

  • CAS Number: 174961-75-2
  • MF: C39H47N3O8S2
  • MW: 749.94
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

H-Arg-OMe.2HCL

H-Arg-OMe.2HCL is an arginine derivative[1].

  • CAS Number: 26340-89-6
  • MF: C7H18Cl2N4O2
  • MW: 261.149
  • Catalog: Others
  • Density: 1.31g/cm3
  • Boiling Point: 329.9ºC at 760 mmHg
  • Melting Point: ~190 °C (dec.)
  • Flash Point: 153.3ºC

D,L-erythro-PDMP hydrochloride

D,L-erythro-PDMP hydrochloride is an erythro isomer of PDMP. D,L-erythro-PDMP hydrochloride causes growth inhibition of cultured rabbit skin fibroblasts. PDMP is an effective inhibitor of UDP-glucose:ceramide glucosyltransferase[1][2].

  • CAS Number: 80943-40-4
  • MF: C23H39ClN2O3
  • MW: 427.02
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Nafocare B1

Nafocare B1 is a synthetic immune biological response modifier.

  • CAS Number: 93135-89-8
  • MF: C11H12O7
  • MW: 256.20900
  • Catalog: Inflammation/Immunology
  • Density: 1.72g/cm3
  • Boiling Point: 332.6ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 154.9ºC

Guanosine 2',3'-Cyclic Phosphate Triethylamine Salt

2′,3′-cGMP triethylamine (Guanosine 2',3'-cyclic phosphate triethylamine) is an active compound. 2′,3′-cGMP triethylamine can be used for various studies[1].

  • CAS Number: 73647-09-3
  • MF: C16H27N6O7P
  • MW: 446.39500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Glutinol acetate

Glutinyl acetate is a triterpene that can be extracted from Dorstenia arifolia. Triterpenes are reported to exhibit anti-inflammatory, antimicrobial, antiviral, cytotoxic and cardiovascular effects[1].

  • CAS Number: 6426-44-4
  • MF: C32H52O2
  • MW: 468.75
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 505.1±29.0 °C at 760 mmHg
  • Melting Point: 192℃ (methanol )
  • Flash Point: 256.2±11.8 °C

Curcumin β-D-Glucuronide

Curcumin-β-D-glucuronide is a major metabolite after oral intake of Curcumin in hepatic tissue and portal blood. Curcumin-β-D-glucuronide can be used for the research of colon cancer[1][2].

  • CAS Number: 227466-72-0
  • MF: C27H28O12
  • MW: 544.50400
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Arzoxifene hydrochloride

Arzoxifene hydrocloride is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue while acting as an estrogen agonist to maintain bone density and lower serum cholesterol.

  • CAS Number: 182133-27-3
  • MF: C28H30ClNO4S
  • MW: 512.060
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: 656.4ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 350.8ºC

Uncargenin C

Uncargenin C is a triterpenoid, which can be isolated from Uncaria rhychophyllo Miq. Jacks. The intermediate of Uncargenin C has anti-leukemia activity, but not itself[1][2].

  • CAS Number: 152243-70-4
  • MF: C30H48O5
  • MW: 488.70
  • Catalog: Cancer
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 621.5±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 343.7±28.0 °C

H-D-Glu-OBzl

H-D-Glu-OBzl is a glutamic acid derivative[1].

  • CAS Number: 79338-14-0
  • MF: C12H15NO4
  • MW: 237.252
  • Catalog: Others
  • Density: 1.245g/cm3
  • Boiling Point: 416.0±40.0 °C at 760 mmHg
  • Melting Point: 154ºC
  • Flash Point: 205.4±27.3 °C

Magnoloside A

Magnoloside A (compound 4) is a main phenylethanoid glycoside in Houpo. Magnoloside A can be used in the research of functional dyspepsia (FD)[1].

  • CAS Number: 113557-95-2
  • MF: C29H36O15
  • MW: 624.59
  • Catalog: Others
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: 908.8±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 294.7±27.8 °C