Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Fmoc-Abg(N3)-OH

Fmoc-Abg(N3)-OH is a click chemistry reagent containing an azide group. Fmoc-Abg(N3)-OH has the potential to synthesize peptide nucleic acids (PNA) and peptoids.

  • CAS Number: 2250433-81-7
  • MF: C21H22N4O4
  • MW: 394.42
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Factor VIIa substrate

Factor VIIa substrate is a colorimetric substrate for Factor VIIa, that can be measured by absorbance at 405 nm[1].

  • CAS Number: 161572-31-2
  • MF: C26H42N8O7S
  • MW: 610.73
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Nα-(2,4-Dinitrophenyl)-L-arginine

Nα-(2,4-Dinitrophenyl)-L-arginine is an arginine derivative[1].

  • CAS Number: 1602-42-2
  • MF: C12H16N6O6
  • MW: 340.29200
  • Catalog: Others
  • Density: 1.65g/cm3
  • Boiling Point: 669.2ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 358.5ºC

SB-633825

SB-633825 is a potent and ATP-competitive inhibitor of TIE2, LOK (STK10) and BRK with IC50s of 3.5 nM, 66 nM, 150 nM, respectively. SB-633825 can inhibit cancer cell growth and angiogenesis[1].

  • CAS Number: 956613-01-7
  • MF: C28H25N3O3S
  • MW: 483.58
  • Catalog: Cardiovascular Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-Bromo-1,1-dichloroacetone

1-Bromo-1,1-dichloroacetone is one of the clorine doxide dsinfection bproducts (DBPs) in drinking water[1].

  • CAS Number: 1751-16-2
  • MF: C3H3BrCl2O
  • MW: 205.86500
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

FGF22-IN-1

FGF22-IN-1 (compound c1) is a potent CD4 D1 inhibitor. FGF22-IN-1 can be used as immunosuppressive agent[1].

  • CAS Number: 113143-13-8
  • MF: C14H11N3OS
  • MW: 269.32
  • Catalog: Inflammation/Immunology
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

N-563

N-563 is an analogue of deoxyspergualin with an immunostimulating activity,it promotes resistance to Candida albicans infection in mice. In vivo: The protective effect of the N-563 against C. albicans infection was investigated in normal and immunosuppressed mice. In normal mice, N-563 treatment at 10 mg/kg for 3 days prior to infection significantly prolonged the survival time. In immunosuppressed mice treated with a single dose of cyclophosphamide 4 days prior to infection, N-563 at 3 and 10 mg/kg for 3 days prior to infection also significantly prolonged the survival time of mice. In addition, it augmented the phagocytic activity of neutrophils and enhanced the delayed type hypersensitivity reaction against C. albicans. Coincidentally, N-563 appeared to protect against secondary infection with C. albicans in the delayed type hypersensitivity-positive mice.[1]N-563 was dissolved in physiological saline and filtered through a Millipore filter (0.22μm).[1]

  • CAS Number: 140686-92-6
  • MF: C15H29N5O5
  • MW: 359.42100
  • Catalog: Others
  • Density: 1.3g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Dactylorhin A

Dactylorhin A, a succinate derivative ester, is isolated from rhizomes of Gymnadenia conopsea. Dactylorhin A exhibits moderate inhibitory effects on NO production effects in RAW 264.7 macrophage cells[1][2].

  • CAS Number: 256459-34-4
  • MF: C40H56O22
  • MW: 888.86
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Pyrromethene 546

BODIPY 493/503 (Pyrromethene 546) is a fluorescent neutral lipid dye (Ex/Em: 493/503 nm). BODIPY 493/503 can facilitate quantification of neutral lipid content by flow cytometry and observation of lipid droplets (LDs) by microscopy[1].

  • CAS Number: 121207-31-6
  • MF: C14H17BF2N2
  • MW: 262.10600
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 257 °C
  • Flash Point: N/A

D-Octamannuronic acid

D-Octamannuronic acid, an alginate oligomer, is produced by marine brown algae and by a limited range of Gram negative bacteria. D-Octamannuronic acid can be used for the research of pain and vascular dementia[1][2][3][4].

  • CAS Number: 862694-98-2
  • MF: C48H66O49
  • MW: 1427.01
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Leflunomide

Leflunomide is a pyrimidine synthesis inhibitor, inhibiting dihydroorotate dehydrogenase, and acts as a disease-modifying antirheumatic drug.

  • CAS Number: 75706-12-6
  • MF: C12H9F3N2O2
  • MW: 270.207
  • Catalog: Cancer
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 289.3±40.0 °C at 760 mmHg
  • Melting Point: 163-168°C
  • Flash Point: 128.8±27.3 °C

Kuguacin R

Kuguacin R is a cucurbitane-type triterpenoid that can be extracted from Momordica charantia L. Kuguacin R possess anti-inflammatory, antimicrobial and anti-viral activities[1].

  • CAS Number: 191097-54-8
  • MF: C30H48O4
  • MW: 472.700
  • Catalog: Infection
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 590.4±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 310.9±30.1 °C

3-Nitrobenzoic acid-d4

3-Nitrobenzoic acid-d4 is the deuterium labeled 3-Nitrobenzoic acid[1].

  • CAS Number: 78399-78-7
  • MF: C7HD4NO4
  • MW: 171.14400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Furin Inhibitor II trifluoroacetate salt

Hexa-D-arginine is an inhibitor of furin.

  • CAS Number: 673202-67-0
  • MF: C36H75N25O6
  • MW: 954.14500
  • Catalog: Peptides
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Oxytocin antiparallel dimer

Oxytocin antiparallel dimer is the disulfide-bridged homo peptide dimer[1].

  • CAS Number: 20054-93-7
  • MF: C86H132N24O24S4
  • MW: 2014.37
  • Catalog: Endocrinology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Methyl (E)-cinnamate-d5

Methyl (E)-cinnamate-d5 is the deuterium labeled Methyl (E)-cinnamate[1]. Methyl (E)-cinnamate (EMC), a phytochemical constituent isolated from Alpinia katsumadai Hayata, is a natural flavor compound with anti-inflammatory properties. Methyl (E)-cinnamate is widely used in the food and commodity industry[2].

  • CAS Number: 61764-82-7
  • MF: C10H5D5O2
  • MW: 167.21600
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

BOC-D-2-Methylphe

Boc-D-Phe(2-Me)-OH is a phenylalanine derivative[1].

  • CAS Number: 80102-29-0
  • MF: C15H21NO4
  • MW: 279.332
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 442.5±40.0 °C at 760 mmHg
  • Melting Point: 116ºC
  • Flash Point: 221.4±27.3 °C

Alcesefoliside

Alcesefoliside is a flavonoid isolated from Nitraria sibirica Pall, with antioxidant activity[1].

  • CAS Number: 124151-38-8
  • MF: C33H40O20
  • MW: 756.65900
  • Catalog: Others
  • Density: 1.79±0.1 g/cm3(Predicted)
  • Boiling Point: 1090.4±65.0 °C(Predicted)
  • Melting Point: N/A
  • Flash Point: N/A

Pivalic acid-d9

Pivalic acid-d9 is the deuterium labeled Pivalic acid[1].

  • CAS Number: 42983-07-3
  • MF: C5HD9O2
  • MW: 111.18700
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Z-Tyr(Bzl)-OH

Z-Tyr(Bzl)-OH is a tyrosine derivative[1].

  • CAS Number: 16677-29-5
  • MF: C24H23NO5
  • MW: 405.443
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 624.4±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 331.5±31.5 °C

Tiplimotide

Tiplimotide (NBI-5788) is an altered peptide ligand (APL) designed from an immunodominant region (83-99) of the neuroantigen myelin basic protein (MBP). Tiplimotide can selectively reduce the production of inflammatory cytokines by pathogenic T-cells. Tiplimotide can be used for the research of multiple sclerosis (MS)[1][2].

  • CAS Number: 178823-49-9
  • MF: C87H142N24O21
  • MW: 1860.207
  • Catalog: Inflammation/Immunology
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Methyltetrazine-amine hydrochloride

Methyltetrazine-Amine, a tetrazine compound, is used for the site-specific dual functionalization of the resulting bioconjugates[1].

  • CAS Number: 1596117-29-1
  • MF: C10H12ClN5
  • MW: 237.69
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Sweroside

Sweroside, isolated from Lonicera japonica, exhibits cytoprotective, anti-osteoporotic, and hepatoprotective effect[1][2].

  • CAS Number: 14215-86-2
  • MF: C16H22O9
  • MW: 358.341
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 630.3±55.0 °C at 760 mmHg
  • Melting Point: 100 °C
  • Flash Point: 231.8±25.0 °C

Onjisaponin Z

Onjisaponin Z is a natural product isolated from Radix Polygalae.

  • CAS Number: 1078708-72-1
  • MF: C71H106O32
  • MW: 1471.58
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

DL-ALANINOL HYDROCHLORIDE

DL-Alaninol hydrochloride is an alanine derivative[1].

  • CAS Number: 17016-92-1
  • MF: C3H10ClNO
  • MW: 111.57100
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 174.5ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 83.9ºC

ingenol-20-hexadecanoate

Ingenol 20-palmitate (compound 2) is a diterpene that can be found in Euphorbia lath yris[1].

  • CAS Number: 39071-33-5
  • MF: C36H58O6
  • MW: 586.84
  • Catalog: Cancer
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 668.3±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 198.1±25.0 °C

4-tert-Butylphthalic anhydride

5-(tert-Butyl)isobenzofuran-1,3-dione is a intermediate and dye. 5-(tert-Butyl)isobenzofuran-1,3-dione has a synonym of 4-tert-Butylphthalic Anhydride[1].

  • CAS Number: 32703-79-0
  • MF: C12H12O3
  • MW: 204.22200
  • Catalog: Others
  • Density: 1.206 g/cm3
  • Boiling Point: 136 °C / 2mmHg
  • Melting Point: 70-75 °C(lit.)
  • Flash Point: 149.9ºC

2,2'-Dichloro bisphenol a mono-D-glucuronide-d12

2,2'-Dichloro bisphenol a mono-D-glucuronide-d12 is the deuterium labeled 2,2'-Dichloro bisphenol a mono-D-glucuronide[1].

  • CAS Number: 2673270-16-9
  • MF: C21H10D12Cl2O8
  • MW: 485.37
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

boc-4,5-dehydro-leu-oh dcha

Boc-4,5-dehydro-Leu-OH (dicyclohexylammonium) salt is a leucine derivative[1].

  • CAS Number: 87720-54-5
  • MF: C23H42N2O4
  • MW: 410.591
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 365ºC at 760 mmHg
  • Melting Point: 148-153ºC
  • Flash Point: 174.5ºC

Oreptacog alfa

Oreptacog alfa is a recombinant DNA derived human blood coagulation factor VIIa. Oreptacog alfa can be used for the research of hemophilia, congenital factor VII deficiency and Glanzmann's thrombasthenia (GT)[1][2].

  • CAS Number: 1360054-92-7
  • MF:
  • MW:
  • Catalog: Cardiovascular Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A