Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Phenylethyl β-D-galactopyranoside

2-Phenylethyl β-D-galactopyranoside (Phenethyl β-D-galactoside) can be synthesized catalyzed by Aspergillus oryzae β-galactosidase[1].

  • CAS Number: 14861-16-6
  • MF: C14H20O6
  • MW: 284.30500
  • Catalog: Others
  • Density: 1.36g/cm3
  • Boiling Point: 486.8ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 248.2ºC

kojic acid

Kojic acid is a natural substance produced by Aspergillus oryzae, also used as an anti-oxidant and radio-protective agent[1].

  • CAS Number: 501-30-4
  • MF: C6H6O4
  • MW: 142.11
  • Catalog: Infection
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 401.7±45.0 °C at 760 mmHg
  • Melting Point: 152-155 °C(lit.)
  • Flash Point: 179.9±22.2 °C

FMRF

FMRF is a peptide consisting of 4 amino acid residues.

  • CAS Number: 74012-06-9
  • MF: C29H41N7O5S
  • MW: 599.74500
  • Catalog: Peptides
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Propacetamol HCl

Propacetamol hydrochloride is an analgesic agent. Propacetamol hydrochloride also is a precursor form of paracetamol. Propacetamol hydrochloride can be used in postoperative pain, acute trauma and gastrointestinal disorders[1].

  • CAS Number: 66532-86-3
  • MF: C14H21ClN2O3
  • MW: 300.781
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: 434.5ºC at 760 mmHg
  • Melting Point: 224-227ºC
  • Flash Point: 216.6ºC

Tesnatilimab

Tesnatilimab is a human IgG4 monoclonal antibody that acts on the immune activating receptor NKG2D and has potential immunomodulatory and anti-inflammatory activity. Tesnatilimab can be used in the study of inflammatory bowel disease (IBD)[1].

  • CAS Number: 2242758-08-1
  • MF:
  • MW:
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-Ser(tBu)-OH

Fmoc-Ser(tBu)-OH is a serine derivative[1].

  • CAS Number: 71989-33-8
  • MF: C22H25NO5
  • MW: 383.438
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 578.6±50.0 °C at 760 mmHg
  • Melting Point: 130.5-135.5 °C(lit.)
  • Flash Point: 303.7±30.1 °C

Fmoc-D-Met-OH

(((9H-Fluoren-9-yl)methoxy)carbonyl)-D-methionine is a Methionine (HY-13694) derivative[1].

  • CAS Number: 112883-40-6
  • MF: C20H21NO4S
  • MW: 371.450
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 614.6±55.0 °C at 760 mmHg
  • Melting Point: 132ºC
  • Flash Point: 325.5±31.5 °C

ACTH (11-24)

ACTH (11-24) is a fragment of adrenocorticotrophin, acts as an antagonist of adrenocorticotropic hormone (ACTH) receptor, and induces cortisol release.

  • CAS Number: 4237-93-8
  • MF: C77H134N24O16
  • MW: 1652.04
  • Catalog: Peptides
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

3,4,5-Trichlorocatechol

3,4,5-Trichlorocatechol is a is a catechol derivative of pentachlorophenol and induces oxidative DNA lesions[1].

  • CAS Number: 56961-20-7
  • MF: C6H3Cl3O2
  • MW: 213.446
  • Catalog: Others
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: 306.5±37.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 139.2±26.5 °C

Terretonin A

Terretonin A is a meroterpenoid that can be isolated from the endophytic fungus Aspergillus terreus[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

4',4'''-Di-O-methylcupressuflavone

4',4'''-Di-O-methylcupressuflavone can be isolated from Phyllanthus sellmianus[1].

  • CAS Number: 74336-91-7
  • MF: C32H22O10
  • MW: 566.511
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: 866.6±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 288.2±27.8 °C

GRK2i

GRK2i is a GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. GRK2i corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.

  • CAS Number: 148505-03-7
  • MF: C153H256N50O41S
  • MW: 3484.045
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Prenylpiperitol

(+)-Piperitol-3,3-dimethylallyl ether can be isolated from the roots and the bark of Zanthoxylum usambarense[1].

  • CAS Number: 157659-20-6
  • MF: C25H28O6
  • MW: 424.49
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 554.7±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 222.7±30.0 °C

S-Fukinolide

Bakkenolide D is the main component of bakkenolide in Petasites tricholobus. Bakkenolide has anti-allergic effects and can be used in the study of allergic rhinitis[1].

  • CAS Number: 18456-03-6
  • MF: C21H28O6S
  • MW: 408.51
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 200-201℃
  • Flash Point: N/A

Atocalcitol

Atocalcitol, a vitamin D3 analogue, is used in the study for psoriasis[1].

  • CAS Number: 302904-82-1
  • MF: C32H46O4
  • MW: 494.70500
  • Catalog: Inflammation/Immunology
  • Density: 1.12g/cm3
  • Boiling Point: 636.3ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 338.6ºC

Arg-Gly-Tyr-Ser-Leu-Gly

Arg-Gly-Tyr-Ser-Leu-Gly is corresponding to the sequence of residues from 21 through 26 in lysozyme. Arg-Gly-Tyr-Ser-Leu-Gly can be used as a substrate for the protein kinase, and phosphorylated at serine residue by protein kinase[1].

  • CAS Number: 59587-18-7
  • MF: C28H45N9O9
  • MW: 651.71200
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Tisagenlecleucel

Tisagenlecleucel (CTL019) is an autologous anti-CD19 chimeric antigen receptor (CAR) T-cell therapy. Tisagenlecleucel targets and eliminates CD19-expressing B cells. Tisagenlecleucel can be used for the research of refractory aggressive diffuse large B-cell lymphoma[1][2].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Yuanhuanin

Yuanhuanin is a natural product that originally recognized in D. sericea. Yuanhuanin also can be isolated also from D. koreana and D. pedunculata[1].

  • CAS Number: 83133-14-6
  • MF: C22H22O11
  • MW: 462.40
  • Catalog: Others
  • Density: 1.609±0.06 g/cm3(Predicted)
  • Boiling Point: 817.5±65.0 °C(Predicted)
  • Melting Point: N/A
  • Flash Point: N/A

Rediocide A

Rediocide A is a highly modified daphnane with potent insecticidal activity. Rediocide A can be isolated from Trigonostemon reidioides[1].

  • CAS Number: 280565-85-7
  • MF: C44H58O13
  • MW: 794.924
  • Catalog: Infection
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Epinodosinol

Epinodosinol is a diterpenoid derived from plant Rabdosia angustifolia. Epinodosinol has inhibitory activity against certain cancer cells[1].

  • CAS Number: 27548-88-5
  • MF: C20H28O6
  • MW: 364.43300
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Anwuweizonic acid

Anwuweizonic acid is a natural compound, isolated from Schisandra propinqua. Anwuweizonic acid is the putative anticancer active principle of Schisandra propinqua[1].

  • CAS Number: 117020-59-4
  • MF: C30H46O3
  • MW: 454.68400
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Pentifylline

Pentifylline is a vasodilator. Pentifylline inhibits platelet aggregation and thromboxane A2 synthesis, decrease the release of free radicals. Pentifylline has the potential for the research of acute ischaemic stroke[1].

  • CAS Number: 1028-33-7
  • MF: C13H20N4O2
  • MW: 264.32300
  • Catalog: Cardiovascular Disease
  • Density: 1.23g/cm3
  • Boiling Point: 452.5ºC at 760mmHg
  • Melting Point: 80-81°C
  • Flash Point: 227.5ºC

Miglitol-d4

Miglitol-d4 is deuterium labeled Miglitol.

  • CAS Number: 2714473-10-4
  • MF: C8H13D4NO5
  • MW: 211.25
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Trioctylamine-d6

Trioctylamine-d6 is the deuterium labeled Trioctylamine[1].

  • CAS Number: 1219798-90-9
  • MF: C24H45D6N
  • MW: 359.71
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Officinalisnin-II

Officinalisnin-II is a natural saponin found in the roots of Asparagus filicinus[1].

  • CAS Number: 57944-19-1
  • MF: C50H84O23
  • MW: 1053.19
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

PI5P4Kα-IN-1

PI5P4Kα-IN-1 (Compound 13) is a PI5P4Kinhibitor (IC50: 2 and 9.4 μM for PI5P4Kα and PI5P4Kβ). PI5P4Kα-IN-1 can be used for research of cancer, metabolic and immunological disorders[1].

  • CAS Number: 2428737-31-7
  • MF: C20H17N3O2S
  • MW: 363.43
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1,2-DIPHYTANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE

DPyPE is a phosphatidylethanolamine lipid composed of polyisoprene alkyl chains. DPyPE is a co-lipid forvaxfectin mixed with GAP-DMORIE in a 1:1 ratio[1].

  • CAS Number: 201036-16-0
  • MF: C45H90NO8P
  • MW: 804.17
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 774.3±70.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 422.1±35.7 °C

7-O-Methylmorroniside

7β-O-Methylmorroniside (7R-O-methylmorroniside) is a R-isomer of 7-O-Methyl morroniside[1].

  • CAS Number: 119943-46-3
  • MF: C18H28O11
  • MW: 420.41
  • Catalog: Others
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 604.5±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 211.8±25.0 °C

Ryuvidine

Ryuvidine is a potent inhibitor of SET domain-containing protein 8(SETD8) with an IC50 of 0.5 µM and suppresses monomethylation of H4K20 in vitro[1]. Ryuvidine also inhibits CDK4 with an IC50 of 6.0 μM and is cytotoxic against a range of human cancer cells[2].

  • CAS Number: 265312-55-8
  • MF: C15H12N2O2S
  • MW: 284.33300
  • Catalog: CDK
  • Density: 1.416g/cm3
  • Boiling Point: 463.8ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 234.3ºC

H-Thr-Pro-OH

H-Thr-Pro-OH is a biologically active peptide.

  • CAS Number: 46398-79-2
  • MF: C9H16N2O4
  • MW: 216.23400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A