Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Oleoyl coenzyme A lithium salt

Oleoyl coenzyme A (Oleoyl-CoA) lithium is a thioester of oleic acid and coenzyme A. Oleoyl coenzyme A lithium has a role as an Escherichia coli metabolite and a mouse metabolite[1][2].

  • CAS Number: 188824-37-5
  • MF: C39H64Li4N7O17P3S
  • MW: 1055.71000
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Secologansaeure

Secologanate is a natural secoiridoid glucoside found in Lonicerae Japonicae Caulis[1].

  • CAS Number: 22864-93-3
  • MF: C16H22O10
  • MW: 374.34000
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

(2H8)Dibenzo[b,d]thiophene

Dibenzothiophene-d8 is the deuterium labeled Dibenzothiophene[1].

  • CAS Number: 33262-29-2
  • MF: C12D8S
  • MW: 192.306
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 332.5±11.0 °C at 760 mmHg
  • Melting Point: 97-100ºC(lit.)
  • Flash Point: 114.8±5.5 °C

11-Azidoundecanoic acid

11-Azidoundecanoic acid is a click chemistry reagent containing an azide group. 11-Azidoundecanoic acid acts as a hydrophobic bioconjugation linker that can be further modified at the azido-position using Staudinger ligation or Click-chemistry. 11-Azidoundecanoic acid is substrate of lipoic acid ligase (LpIA) for labeling[1][2].

  • CAS Number: 118162-45-1
  • MF: C11H21N3O2
  • MW: 227.30300
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

3,3',4,4'-Biphenyltetramine tetrahydrochloride

3,3'-Diaminobenzidine(DAB) is an organic compound that is both chemically and thermodynamically stable; DAB has been used in immunohistochemical staining of nucleic acids and proteins.

  • CAS Number: 7411-49-6
  • MF: C12H18Cl4N4
  • MW: 360.110
  • Catalog: Dye Reagents
  • Density: N/A
  • Boiling Point: 481.7ºC at 760 mmHg
  • Melting Point: 300°C
  • Flash Point: 282.7ºC

Alitame

Alitame (anhydrous) is a high-intensity sweetener formed from the amino acids L-aspartic acid and D-alanine, and an amine derived from thietane[1].

  • CAS Number: 80863-62-3
  • MF: C14H25N3O4S
  • MW: 331.43
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 608.5±55.0 °C at 760 mmHg
  • Melting Point: 136-147°
  • Flash Point: 321.8±31.5 °C

Tiliquinol

Tiliquinol (NSC 130828) is a non-absorbed anti-amoebic luminal agent. Tiliquinol is used in combination with tibroquinol. Tiliquinol can be used for the research of amebic liver abscess[1][2].

  • CAS Number: 5541-67-3
  • MF: C10H9NO
  • MW: 159.185
  • Catalog: Infection
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 324.7±22.0 °C at 760 mmHg
  • Melting Point: 122-124°C
  • Flash Point: 150.2±22.3 °C

Difloxacin-d3 hydrochloride

Difloxacin-d3 (hydrochloride) is the deuterium labeled Difloxacin (hydrochloride)[1].

  • CAS Number: 1173021-89-0
  • MF: C21H17D3ClF2N3O3
  • MW: 438.87
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Schisanlignone D

Schisanlignone D is a chemical component of Schisandra viridis a. c. sm[1].

  • CAS Number: 144606-84-8
  • MF: C22H22O7
  • MW: 398.406
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 593.5±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 259.7±30.2 °C

Z-LYS-SBZL HCL

Z-LYS-SBZL (monohydrochloride) is a lysine derivative[1].

  • CAS Number: 69861-89-8
  • MF: C21H27ClN2O3S
  • MW: 422.96900
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 566.3ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 296.3ºC

Wilfordinine D

Wilfordinine D is a natural sesquiterpene alkaloid[1].

  • CAS Number: 256937-98-1
  • MF: C41H47NO19
  • MW: 857.81
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

S-(4-nitrophenyl)-L-cysteine

S-(4-Nitrophenyl)-L-cysteine is a cysteine derivative[1].

  • CAS Number: 55288-30-7
  • MF: C9H10N2O4S
  • MW: 242.25200
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

JJH260

JJH260 is AIG1inhibitor, and inhibit the fluorophosphonate reactivity and fatty acid esters of hydroxy fatty acid (FAHFA) hydrolysis activity of AIG1in HEK293T cells, with IC50 values of 0.50 μM and 0.57 μM, respectively[1].

  • CAS Number: 1831135-30-8
  • MF: C29H34ClN5O5
  • MW: 568.06
  • Catalog: MAGL
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 703.9±70.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 379.5±35.7 °C

ISIS 416858

ISIS 416858, a single-stranded antisense oligodeoxynucleotide, is a potent and selective inhibitor of FXI mRNA expression.

  • CAS Number: 1223657-78-0
  • MF:
  • MW:
  • Catalog: Cardiovascular Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-Gln(Trt)-Ser(psi(Me,Me)pro)-OH

Fmoc-Gln(Trt)-Ser(psi(Me,Me)pro)-OH is a dipeptide.

  • CAS Number: 1821378-64-6
  • MF: C45H43N3O7
  • MW: 737.839
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 974.6±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 543.2±34.3 °C

BI-0115

BI-0115 is a selective inhibitor of LOX-1 (IC50=5.4 µM) that blocks cellular uptake of oxLDL. BI-0115 binding triggers receptor inhibition by formation of dimers of the homodimeric ligand binding domain[1].

  • CAS Number: 4929-23-1
  • MF: C15H14ClN3O
  • MW: 287.744
  • Catalog: Cardiovascular Disease
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 489.2±45.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 249.7±28.7 °C

Dibromo(chloro)nitromethane

Dibromochloronitromethane is one of Halonitromethanes, which are a recently identified class of disinfection by-products (DBPs) in drinking water[1].

  • CAS Number: 1184-89-0
  • MF: CBr2ClNO2
  • MW: 253.277
  • Catalog: Others
  • Density: 2.6±0.1 g/cm3
  • Boiling Point: 134.9±35.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 35.4±25.9 °C

Muramic acid

Muramic acid is a component in many Gram-positive bacterial cell walls, as marker for Gram-positive bacteria[1].

  • CAS Number: 1114-41-6
  • MF: C9H17NO7
  • MW: 251.23400
  • Catalog: Others
  • Density: 1.51 g/cm3
  • Boiling Point: 572.4ºC at 760 mmHg
  • Melting Point: 140-150 °C (dec.)
  • Flash Point: 300ºC

Desmethyl-WEHI-345 analog

Desmethyl-WEHI-345 analog is a protein kinase inhibitor extracted from patent WO2012003544A1, example 12. Desmethyl-WEHI-345 analog can be used for the research of colon cancer[1].

  • CAS Number: 1354825-03-8
  • MF: C22H23N7O
  • MW: 401.46
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

BODIPY FL Thapsigargin

BODIPY FL Thapsigargin is a potent green fluorescent dye. BODIPY FL Thapsigargin inhibits intracellular SERCA-type Ca2+ pumps present in the sarcoplasmic/endoplasmic reticulum. BODIPY FL Thapsigargin used for investigation of thapsigargin binding sites in live cells[1][2].

  • CAS Number: 216571-99-2
  • MF: C44H57B3F2N2O122-
  • MW: 876.36
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

7-[[2-O-(6-deoxy-alpha-L-mannopyranosyl)-beta-D-glucopyranosyl]oxy]-3,5-dihydroxy-2-(4-hydroxyphenyl)-4H-benzopyran-4-one

Kaempferol 7-O-neohesperidoside is a ?avonoid glycoside that can be isolated from Litchi chinensis. Kaempferol 7-O-neohesperidoside exhibits significant cytotoxic activity against A549, LAC, Hep-G2, and HeLa cell lines with IC50s of 0.53, 7.93, 0.020, and 0.051 μM, respectively[1].

  • CAS Number: 17353-03-6
  • MF: C27H30O15
  • MW: 594.51800
  • Catalog: Cancer
  • Density: 1.76g/cm3
  • Boiling Point: 934.7ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 310.4ºC

3,4-Di-O-acetyl-L-fucal

3,4-Di-O-acetyl-L-fucal is the reactant for synthesis antibiotics (extracted from patent WO1999026956A1)[1].

  • CAS Number: 54621-94-2
  • MF: C10H14O5
  • MW: 214.21500
  • Catalog: Others
  • Density: 1.16g/cm3
  • Boiling Point: 295.9ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 116.5ºC

Metopimazine

Metopimazine (EXP999) is a phenothiazine derivative used to prevent emesis during chemotherapy. Metopimazine belongs to the anti-dopaminergic anti-emetics (ADA) class. Metopimazine can be used for the research of gastroenteritis (GE) [1].

  • CAS Number: 14008-44-7
  • MF: C22H27N3O3S2
  • MW: 445.598
  • Catalog: Inflammation/Immunology
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 679.0±65.0 °C at 760 mmHg
  • Melting Point: 170.5℃
  • Flash Point: 364.4±34.3 °C
  • CAS Number: 415684-38-7
  • MF: C62H93N19O23
  • MW: 1472.515
  • Catalog: Others
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Endoxifen (hydrochloride)

Endoxifen hydrochloride, the active metabolite of Tamoxifen, is a potent antiestrogen that targets estrogen receptor.

  • CAS Number: 1197194-41-4
  • MF: C25H28ClNO2
  • MW: 409.948
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Quercetin 3-O-malonylglucoside

Quercetin 3-O-(6''-O-malonyl)-β-D-glucoside, a natural flavonol glycoside, possesses antioxidant activity[1].

  • CAS Number: 96862-01-0
  • MF: C24H22O15
  • MW: 550.42200
  • Catalog: Metabolic Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 195-201 °C
  • Flash Point: N/A

Pyrimethanil-d5

Pyrimethanil-d5 is the deuterium labeled Hypoxanthine. Hypoxanthine, a purine derivative, is a potential free radical generator and could be used as an indicator of hypoxia.

  • CAS Number: 2118244-83-8
  • MF: C12H8D5N3
  • MW: 204.28
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

DL-Dithiothreitol

DTT is a small-molecule redox reagent.

  • CAS Number: 3483-12-3
  • MF: C4H10O2S2
  • MW: 154.251
  • Catalog: Biochemical Assay Reagents
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 364.5±42.0 °C at 760 mmHg
  • Melting Point: 38-43ºC
  • Flash Point: 174.2±27.9 °C

Polyporoid B

Polyporoid B is a ergostane-type ecdysteroid that exhibits potent anti-inflammatory activity in vivo[1].

  • CAS Number: 1042362-45-7
  • MF: C28H44O7
  • MW: 492.64
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

DL-Panthenol

DL-Panthenol is an intermediate of organic synthesis.

  • CAS Number: 16485-10-2
  • MF: C9H19NO4
  • MW: 205.251
  • Catalog: Biochemical Assay Reagents
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 483.6±45.0 °C at 760 mmHg
  • Melting Point: 66-69 °C(lit.)
  • Flash Point: 246.3±28.7 °C