An antifungal agent is a drug that selectively eliminates fungal pathogens from a host with minimal toxicity to the host. Classes: 1. Polyene Antifungal Drugs: Amphotericin, nystatin, and pimaricin interact with sterols in the cell membrane (ergosterol in fungi, cholesterol in humans) to form channels through which small molecules leak from the inside of the fungal cell to the outside. 2. Azole Antifungal Drugs: Fluconazole, itraconazole, and ketoconazole inhibit cytochrome P450-dependent enzymes (particularly C14-demethylase) involved in the biosynthesis of ergosterol, which is required for fungal cell membrane structure and function. 3. Allylamine and Morpholine Antifungal Drugs: lylamines (naftifine, terbinafine) inhibit ergosterol biosynthesis at the level of squalene epoxidase. The morpholine drug, amorolfine, inhibits the same pathway at a later step. 4. Antimetabolite Antifungal Drugs: 5-Fluorocytosine acts as an inhibitor of both DNA and RNA synthesis via the intracytoplasmic conversion of 5-fluorocytosine to 5-fluorouracil.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
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Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
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Epigenetics >
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JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
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Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
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Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
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Protein Tyrosine Kinase/RTK >
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Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
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Vitamin D Related >
VD/VDR
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Antimicrobial agent-3

Antimicrobial agent-3 (Compound U10) is an antimicrobial agent against bacterial, fungal and tubercular infections[1].

  • CAS Number: 1902712-34-8
  • MF: C14H11N3OS
  • MW: 269.32
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Aleurodiscal

Aleurodiscal is an fungal inhibitor that can be obtained from cultures of Aleurodiscus mirabilis. Aleurodiscal can be used in the study of fungal infections[1].

  • CAS Number: 122535-46-0
  • MF: C30H46O6
  • MW: 502.68300
  • Catalog: Fungal
  • Density: 1.19g/cm3
  • Boiling Point: 642.5ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 204ºC

Isoprothiolane

Isoprothiolane is a systemic fungicide. Isoprothiolane is a rice blast controlling agent against the fungal disease of rice planty Pyvioutavia oryzae Cav[1].

  • CAS Number: 50512-35-1
  • MF: C12H18O4S2
  • MW: 290.39900
  • Catalog: Fungal
  • Density: 1.228 g/cm3
  • Boiling Point: 353ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 159ºC

Dermaseptin-S2

Dermaseptin-S2 is an antimicrobial peptide derived from frog skin against filamentous fungi[1].

  • CAS Number: 151896-13-8
  • MF: C155H255N43O43S2
  • MW: 3473.08
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Triclosan D3

Triclosan D3 is the deuterium labeled Triclosan. Triclosan is an antibacterial and antifungal agent found in consumer products, including soaps, detergents, toys, and surgical cleaning treatments[1][2].

  • CAS Number: 1020719-98-5
  • MF: C12H7Cl3O2
  • MW: 289.54200
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Xanthobaccin A

Xanthobaccin A is an antifungal compound, can be isolated from the culture fluid of Stenotrophomonas sp. strain SB-K88. Xanthobaccin A has potent inhibitory effect on sugar beet damping-off disease[1][2][3].

  • CAS Number: 227596-81-8
  • MF: C29H38N2O6
  • MW: 510.622
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 819.4±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 449.4±34.3 °C

Loflucarban

Loflucarban (Fluonilid) is a potent antimycotic agent. Loflucarban can be used for the research of the ear infections[1].

  • CAS Number: 790-69-2
  • MF: C13H9Cl2FN2S
  • MW: 315.19300
  • Catalog: Fungal
  • Density: 1.531g/cm3
  • Boiling Point: 395ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 192.7ºC

ChloraMultilide B

Chloramultilide B is a lindenane dimer that can be isolated from Chloranthus serratus. Chloramultilide B has inhibitory activities against Candida albicans and C.parapsilosis with a MIC value of 0.068 μM[1].

  • CAS Number: 1000995-47-0
  • MF: C39H42O14
  • MW: 734.742
  • Catalog: Fungal
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

4-Amino-2-methyl-1-naphthol

Vitamin K5 (Synkamin) is a photosensitizer and a antimicrobial agent. Vitamin K5 is a specific PKM2 inhibitor with IC50 values of 28, 191 and 120 μM for PKM2, PKM1 and PKL. Vitamin K5 induces apoptosis of colon 26 cells. Vitamin K5 can be used for the research of infection and cancer, and it also can be used as a preservative for pharmaceuticals, foods, and beverages[1][2][3].

  • CAS Number: 83-70-5
  • MF: C11H11NO
  • MW: 173.211
  • Catalog: Bacterial
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 385.1±30.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 186.7±24.6 °C

Tetramethylkaempferol

Tetramethylkaempferol is an antifungal agent. Tetramethylkaempferol shows antifungal activity against Candida albicansCandida albicans with an IC50 value of 17.63 µg/mL[1].

  • CAS Number: 16692-52-7
  • MF: C19H18O6
  • MW: 342.34
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 540.6±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 239.2±30.2 °C

Sulconazole mononitrate

Sulconazole mononitrate ((±)-Sulconazole mononitrate), an imidazole derivative, is a broad-spectrum fungicide and is inhibitory to certain gram-positive anaerobes. Sulconazole mononitrate can be used for the research of dermatomycoses, pityriasis versicolor, and cutaneous candidiasis[1][2].

  • CAS Number: 61318-91-0
  • MF: C18H16Cl3N3O3S
  • MW: 460.76200
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: 558.2ºC at 760 mmHg
  • Melting Point: 130.5-132℃
  • Flash Point: 291.4ºC

Valtrate Hydrine B4

Valtrate hydrine B4 is a natural compound with antifungal activities[1].

  • CAS Number: 18296-48-5
  • MF: C27H40O10
  • MW: 524.60000
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

rabdoserrin A

Rabdoserrin A is a diterpenoid. Rabdoserrin A has antifungal activity[1][2].

  • CAS Number: 96685-01-7
  • MF: C20H26O5
  • MW: 346.41700
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Butenafine

Butenafine is a potent and broad spectrum benzylamine antifungal agent[1]. Butenafine inhibits fungal ergosterol biosynthesis at the point of squalene epoxidation, leading to a deficiency of the fungal cell membranes. Butenafine is effective against dermatophytes infections, such as  tinea pedis,  tinea cruris, tinea versicolor[1][2].

  • CAS Number: 101828-21-1
  • MF: C23H27N
  • MW: 317.467
  • Catalog: Fungal
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 426.1±14.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 187.7±17.0 °C

Nikkomycin Z

Nikkomycin Z, a nucleoside-peptide, is a selective competitive chitin synthesis inhibitor. Nikkomycin Z has antifungal effects and acts as a competitive analogue of the chitin synthase substrate UDP-N-acetylglucosamine[1].

  • CAS Number: 59456-70-1
  • MF: C20H25N5O10
  • MW: 495.44000
  • Catalog: Fungal
  • Density: 1.646 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

verazine

Verazine ((-)-Verazine) is an anti-Fungal Agent that can be found in the dried roots and rhizoma of Veratrum maackii Regel. Verazine causes DNA damage in the cerebellum and cerebral cortex of mice in a dose-dependent manner. Verazine can be used in the study of fungal infections and neurological diseases[1][2].

  • CAS Number: 14320-81-1
  • MF: C27H43NO
  • MW: 397.64
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

famoxadone

Famoxadone (DPX-JE874) is a fungicide acting against a broad spectrum of fungi and is widely used in Integrated Pest Management strategies in different agricultural crops[1].

  • CAS Number: 131807-57-3
  • MF: C22H18N2O4
  • MW: 374.389
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 491.3±55.0 °C at 760 mmHg
  • Melting Point: 140.3-141.8ºC
  • Flash Point: 250.9±31.5 °C

Epoxiconazole

Epoxiconazole, a fungicide, is a demethylation inhibitor of the Ergosterol biosynthesis pathway. Epoxiconazole exhibits strong inhibitory effects on both carbendazim-resistant and phenamacril-resistant isolates, and can be used for controlling many crop diseases[1].

  • CAS Number: 133855-98-8
  • MF: C17H13ClFN3O
  • MW: 329.756
  • Catalog: Fungal
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 463.1±55.0 °C at 760 mmHg
  • Melting Point: 125°C (lit.)
  • Flash Point: 233.9±31.5 °C

Debneyol

Debneyol exhibits more potent fungicidal activity than validamycin.

  • CAS Number: 99694-82-3
  • MF: C15H26O2
  • MW: 238.37
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Abafungin

Abafungin, a antifungal agent, inhibitis the transmethylation at the C-24 position of the sterol side chain, catalyzed by the enzyme sterol-C-24-methyltransferase.

  • CAS Number: 129639-79-8
  • MF: C21H22N4OS
  • MW: 378.491
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 533.6±52.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 276.5±30.7 °C

ASP2397

ASP2397 (VL-2397), a natural compound, exhibits rapid and potent fungicidal activity against Aspergillus species, at a MIC range of 1 to 4 μg/mL in human serum. ASP2397 (VL-2397) has the potential to treat invasive pulmonary aspergillosis (IPA)[1].

  • CAS Number: 2088622-19-7
  • MF: C40H59AlN10O13
  • MW: 914.94
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Herbicidin A

Herbicidin A is an adenosine-derived nucleoside antibiotic, but also is a herbicide against dicotyledonous plants. Herbicidin A can be isolated from Streptomyces scopuliridis M40[1][2].

  • CAS Number: 55353-31-6
  • MF: C23H29N5O11
  • MW: 551.50300
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

pyrimorph

Pyrimorph is a fungicide with excellent antifungal activity against oomycetes[1].

  • CAS Number: 868390-90-3
  • MF: C22H25ClN2O2
  • MW: 384.90
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 131-133 °C
  • Flash Point: N/A

Caffeic Acid-13C3

Caffeic acid-13C3 (3,4-Dihydroxycinnamic acid-13C3) is an 13C labeled caffeic acid. Caffeic acid is a phytonutrient belonging to the flavonoids. Caffeic acid and its derivatives, are potential antimicrobial agents, chronic infection induced by microbes such as bacteria, fungi, and viruses[1].

  • CAS Number: 1185245-82-2
  • MF: C613C3H8O4
  • MW: 183
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 223-225°C (dec.)
  • Flash Point: N/A

Dermaseptin-S3

Dermaseptin-S3 is an antimicrobial peptide derived from frog skin against filamentous fungi[1].

  • CAS Number: 151896-14-9
  • MF: C138H240N38O35S
  • MW: 3023.68
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

2-Furancarboxaldehyde,5-nitro-, oxime, [C(Z)]-

Nifuroxime is an anti-infective agent. Nifuroxime can be used in the research of fungal infections[1].

  • CAS Number: 6236-05-1
  • MF: C5H4N2O4
  • MW: 156.09600
  • Catalog: Fungal
  • Density: 1.58g/cm3
  • Boiling Point: 274.8ºC at 760 mmHg
  • Melting Point: 160-163ºC
  • Flash Point: 120ºC

Potassium Gluconate

Potassium Gluconate (Potassium D-gluconate) is an orally active carboxylic acid by the oxidation with antiseptic and chelating properties[1].

  • CAS Number: 299-27-4
  • MF: C6H11KO7
  • MW: 234.246
  • Catalog: Fungal
  • Density: 1.73 g/cm3
  • Boiling Point: 673.6ºC at 760 mmHg
  • Melting Point: 183 °C (dec.)(lit.)
  • Flash Point: 375.2ºC

Fluxapyroxad

Fluxapyroxad is a synthetic broad-spectrum fungicide for the control of fungal diseases. It works by inhibiting succinate dehydrogenase in complex II of the mitochondrial respiratory chain, resulting in inhibition of spore germination, germ tubes and mycelia growth within the fungus target species[1].

  • CAS Number: 907204-31-3
  • MF: C18H12F5N3O
  • MW: 381.30
  • Catalog: Fungal
  • Density: 1.42g/cm3
  • Boiling Point: 428.4ºC at 760 mmHg
  • Melting Point: 156.8 ℃
  • Flash Point: 212.9ºC

(+)-Magnoflorine chloride

Magnoflorine chloride (Magnoflorine chloride), an aporphine alkaloid found in Acoruscalamus, reduces the formation of C. albicans biofilm[1]. Magnoflorine chloride has anti-fungal, anti-antidiabetic and anti-oxidative activity[2].

  • CAS Number: 6681-18-1
  • MF: C20H24ClNO4
  • MW: 377.862
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

APX001

APX001 (APX 001A;E1210) is a novel broad-spectrum antifungal agent that inhibits the fungal protein Gwt1, demonstrates significantly acitive MIC50 and MIC90 values of 0.004 and 0.031 ug/ml (16 strains of C. auris); inhibits the inositol acylation activity of C. albicans Gwt1p and A. fumigatus Gwt1p with IC50 of 0.3 to 0.6 uM but has no inhibitory activity against human Pig-Wp; shows significant efficacy in murine model of disseminated C. auris infection, and log reduction in CFU counts in kidney, lung, and brain tissue. Fungal Infection Phase 1 Clinical

  • CAS Number: 936339-60-5
  • MF: C21H18N4O2
  • MW: 358.393
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 569.4±45.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 298.1±28.7 °C