An antifungal agent is a drug that selectively eliminates fungal pathogens from a host with minimal toxicity to the host. Classes: 1. Polyene Antifungal Drugs: Amphotericin, nystatin, and pimaricin interact with sterols in the cell membrane (ergosterol in fungi, cholesterol in humans) to form channels through which small molecules leak from the inside of the fungal cell to the outside. 2. Azole Antifungal Drugs: Fluconazole, itraconazole, and ketoconazole inhibit cytochrome P450-dependent enzymes (particularly C14-demethylase) involved in the biosynthesis of ergosterol, which is required for fungal cell membrane structure and function. 3. Allylamine and Morpholine Antifungal Drugs: lylamines (naftifine, terbinafine) inhibit ergosterol biosynthesis at the level of squalene epoxidase. The morpholine drug, amorolfine, inhibits the same pathway at a later step. 4. Antimetabolite Antifungal Drugs: 5-Fluorocytosine acts as an inhibitor of both DNA and RNA synthesis via the intracytoplasmic conversion of 5-fluorocytosine to 5-fluorouracil.


Anti-infection >
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NF-κB >
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Vitamin D Related >
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Esculentoside B

Esculentoside B (Phytolaccoside B) is a natural product from the roots of Phytolacca acinosa Roxb. Esculentoside B is neurotoxic to zebrafish larvae, and impairs their central nervous system development. Esculentoside B inhibits inflammatory response and has antifungal activity[1][2][3].

  • CAS Number: 60820-94-2
  • MF: C36H56O11
  • MW: 664.82
  • Catalog: Fungal
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 779.3±60.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 237.0±26.4 °C

Ethacridine lactate Monohydrate

Ethacridine lactate monohydrate is an aromatic organic compound, primarily use as an antiseptic.

  • CAS Number: 6402-23-9
  • MF: C18H23N3O5
  • MW: 361.392
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: 523.5ºC at 760 mmHg
  • Melting Point: 243-245 °C(lit.)
  • Flash Point: 270.4ºC

Griseofulvin

Griseofulvin(Gris-PEG; Grifulvin) is a spirocyclic fungal natural product used in treatment of fungal dermatophytes; Antifungal drug.

  • CAS Number: 126-07-8
  • MF: C17H17ClO6
  • MW: 352.766
  • Catalog: Fungal
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 570.4±50.0 °C at 760 mmHg
  • Melting Point: 218-220 °C(lit.)
  • Flash Point: 228.0±29.1 °C

SDH-IN-3

SDH-IN-3 is a succinate dehydrogenase (SDH) inhibitor with an IC50 of 7.2 μg/mL. SDH-IN-3 exhibits excellent antifungal activities against Nigrospora oryzae with an EC50 of 1.9 μg/mL. SDH-IN-3 can be used for anti-infection research[1].

  • CAS Number: 2805297-11-2
  • MF: C15H11F2N3OS
  • MW: 319.33
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Antifungal agent 14

Antifungal agent 14 exhibits broad-spectrum activity against the fungal strains with excellent minimum inhibitory concentration values.

  • CAS Number: 2710259-38-2
  • MF: C18H19N7O3
  • MW: 381.39
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Magnoflorine Iodide

(+)-Magnoflorine iodide (Magnoflorine iodide), an aporphine alkaloid found in Acoruscalamus, reduces the formation of C. albicans biofilm[1]. (+)-Magnoflorine iodide has anti-fungal, anti-antidiabetic and anti-oxidative activity[2].

  • CAS Number: 4277-43-4
  • MF: C20H24INO4
  • MW: 469.31300
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 248-249ºC
  • Flash Point: N/A

Idarubicin

Idarubicin is an orally active and potent anthracycline antileukemic agent. Idarubicin inhibits the topoisomerase II interfering with the replication of DNA and RNA transcription. Idarubicin shows induction of DNA damage. Idarubicin inhibits DNA synthesis and of c-myc expression. Idarubicin inhibits the growth of bacteria and yeasts[1][2][3][4][5].

  • CAS Number: 58957-92-9
  • MF: C26H27NO9
  • MW: 497.494
  • Catalog: Bacterial
  • Density: 1.6±0.1 g/cm3
  • Boiling Point: 725.4±60.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 392.5±32.9 °C

Nystatin

Nystatin is a polyene antifungal antibiotic effective against yeast and mycoplasma.

  • CAS Number: 1400-61-9
  • MF: C47H75NO17
  • MW: 276.414
  • Catalog: Fungal
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 400.2±14.0 °C at 760 mmHg
  • Melting Point: >155°C (dec.)
  • Flash Point: 297.0±15.2 °C

Norbatzelladine L

Norbatzelladine L (Compound 2) is an inhibitor of the catalytic and functional activity of Pdr5p transporter. Norbatzelladine L inhibits Pdr5p ATPase activity with an IC50 of 3.8 µM. Norbatzelladine L shows antifungal, antiparasitic, antiviral, antibacterial and antitumoral activities[1].

  • CAS Number: 1187954-93-3
  • MF: C38H66N6O2
  • MW: 638.97
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Undecanoic acid

Undecanoic acid (Undecanoate) is a monocarboxylic acid with antimycotic property, which inhibits the production of exocellular keratinase, lipase and the biosynthesis of several phospholipids in T. rubrum[1].

  • CAS Number: 112-37-8
  • MF: C11H22O2
  • MW: 186.291
  • Catalog: Fungal
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 283.3±3.0 °C at 760 mmHg
  • Melting Point: 28-31 °C(lit.)
  • Flash Point: 128.2±11.9 °C

BTL peptide

BTL peptide is an antifungal peptide. BTL peptide is active against B. maydis, A. brassicae, A. niger and C. personata[1].

  • CAS Number: 1021461-47-1
  • MF: C67H114N18O24
  • MW: 1555.73
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Triadimenol-d4

Triadimenol-d4 is the deuterium labeled Triadimenol[1]. Triadimenol is a triazole fungicide and has been widely used in agriculture. Triadimenol has certain toxicity to animals[2].

  • CAS Number: 2121989-56-6
  • MF: C14H14D4ClN3O2
  • MW: 299.79
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

benzoic acid

Benzoic Acid is an aromatic alcohol existing naturally in many plants and is a common additive to food, drinks, cosmetics and other products. It acts as preservatives through inhibiting both bacteria and fungi.

  • CAS Number: 65-85-0
  • MF: C7H6O2
  • MW: 122.12
  • Catalog: Bacterial
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 249.3±9.0 °C at 760 mmHg
  • Melting Point: 121-125 °C(lit.)
  • Flash Point: 121.1±0.0 °C

trichodecenin II

Trichodecenin II is a fungal metabolite that can be found in conidia of the fungus, Trichoderma viride[1].

  • CAS Number: 140939-04-4
  • MF: C38H69N7O8
  • MW: 751.99700
  • Catalog: Fungal
  • Density: 1.109g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Xenopsin precursor fragment

Xenopsin precursor fragment is an antimicrobial peptide, and has antibacterial/antifungal (10-500 μg/mL) and anti-protozoal (MIC: 2-20 μg/mL) activity[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

10-Undecenoic acid

10-Undecenoic acid was used as a starting reagent in the syntheses of Pheromone (11Z)-hexadecenal.

  • CAS Number: 112-38-9
  • MF: C11H20O2
  • MW: 184.275
  • Catalog: Fungal
  • Density: 0.9±0.1 g/cm3
  • Boiling Point: 300.8±0.0 °C at 760 mmHg
  • Melting Point: 23-25 °C(lit.)
  • Flash Point: 148.9±0.0 °C

Bronidox

5-Bromo-5-nitro-1,3-dioxane, an antimicrobial compound, is effective against Gram-positive and Gram-negative bacteria and fungi, including yeast. 5-Bromo-5-nitro-1,3-dioxane inhibits enzyme activity and subsequent inhibition of microbial growth by the oxidation of essential protein thiol[1].

  • CAS Number: 30007-47-7
  • MF: C4H6BrNO4
  • MW: 211.999
  • Catalog: Bacterial
  • Density: 1.8±0.1 g/cm3
  • Boiling Point: 280.8±40.0 °C at 760 mmHg
  • Melting Point: 60°C
  • Flash Point: 123.6±27.3 °C

Posaconazole

Posaconazole is a broad-spectrum, second generation, triazole compound with antifungal activity.

  • CAS Number: 171228-49-2
  • MF: C37H42F2N8O4
  • MW: 700.777
  • Catalog: Fungal
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 850.7±75.0 °C at 760 mmHg
  • Melting Point: 170-1720C
  • Flash Point: 468.3±37.1 °C

Methasulfocarb

Methasulfocarb is a fungicide compound.

  • CAS Number: 66952-49-6
  • MF: C9H11NO4S2
  • MW: 261.31800
  • Catalog: Fungal
  • Density: 1.42g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Phosphatase-IN-1

Phosphatase-IN-1 (compound II-8), a propranolol (HY-B0573B) derivative, is a phosphatidate phosphatase (Pah) inhibitor. Phosphatase-IN-1 can binds to MoPah1, with an affinity constant of 19.8 μM. Phosphatase-IN-1 inhibits growth of plant pathogens and shows anti-fungal ability. Phosphatase-IN-1 is not toxic to rice seedlings and wheat heads[1].

  • CAS Number: 2889356-55-0
  • MF: C16H16Cl2FNO2
  • MW: 344.21
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Antifungal agent 49

Antifungal agent 49 (Example 112) is an antifungal agent. Antifungal agent 49 is active against Cryptococcus neoformans with a MIC value of 49 μM[1].

  • CAS Number: 1414861-21-4
  • MF: C15H12O4
  • MW: 256.25
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Sulconazole (nitrate)

Sulconazole nitrate is an antifungal medication of the imidazole class.

  • CAS Number: 82382-23-8
  • MF: C18H15Cl3N2S.HNO3
  • MW: 460.76
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: 558.2ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 291.4ºC

Pradimicin A

Pradimicin A (PRM-A) is a potent antifungal agent, with an MIC of 4 μg/mL against Candida rugosa. Pradimicin A has antiviral activities against CoV, HIV and other enveloped viruses. Pradimicin A shows aggregation property, and can recognize d-Man in the presence of Ca2+ ion[1][2].

  • CAS Number: 117704-65-1
  • MF: C40H44N2O18
  • MW: 840.78
  • Catalog: Fungal
  • Density: 1.688g/cm3
  • Boiling Point: 1120.269°C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 631.316°C

Isobellidifolin

Isobellidifolin, a xanthone, is a free radical scavenger and antioxidant compound. Isobellidifolin has potent antifungal effect[1].

  • CAS Number: 552-00-1
  • MF: C14H10O6
  • MW: 274.22600
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Daidzein dimethyl ether

4',7-Dimethoxyisoflavone is isolated from the leaves of Albizzia lebbeck, which shows antifungal activity.

  • CAS Number: 1157-39-7
  • MF: C17H14O4
  • MW: 282.29100
  • Catalog: Fungal
  • Density: 1.242g/cm3
  • Boiling Point: 452.8ºC at 760mmHg
  • Melting Point: 161-163°C
  • Flash Point: 202.2ºC

Moniliformin, sodium salt

Moniliformin sodium salt is a potent, water-soluble mycotoxin isolate from Fusarium moniliforme.

  • CAS Number: 71376-34-6
  • MF: C4HNaO3
  • MW: 120.03900
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: 239.6ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 113ºC

Undecanoic acid-d2

Undecanoic acid-d2 is the deuterium labeled Undecanoic acid. Undecanoic acid (Undecanoate) is a monocarboxylic acid with antimycotic property, which inhibits the production of exocellular keratinase, lipase and the biosynthesis of several phospholipids in T. rubrum[1].

  • CAS Number: 64118-43-0
  • MF: C11H20D2O2
  • MW: 188.30
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Sodium Houttuyfonate

Sodium Houttuyfonate is a natural compound extracted from Houttuynia cordata, with anti-inflammatory and anti-fibrotic effects. Sodium Houttuyfonate ameliorates LPS induced mastitis by inhibiting the NF κB pathway[1][2].

  • CAS Number: 83766-73-8
  • MF: C12H23NaO5S
  • MW: 302.363
  • Catalog: Bacterial
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Eberconazole nitrate

Eberconazole nitrate is a dichlorinated imidazole derivative with antifungal activity. Eberconazole nitrate is more active than Clotrimazole, Ketoconazole, and Miconazole. Eberconazole nitrate has the potential for the research of dermatophytoses with a topical administration[1].

  • CAS Number: 130104-32-4
  • MF: C18H15Cl2N3O3
  • MW: 392.236
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: 495ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 253.2ºC

Fluopyram

Fluopyram is a succinate dehydrogenase inhibitor fungicide, inhibits the growth of F. virguliforme isolates with mean EC50 of 3.35 µg/mL[1].

  • CAS Number: 658066-35-4
  • MF: C16H11ClF6N2O
  • MW: 396.71
  • Catalog: Fungal
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A