Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

Anilofos

Anilofos is a pre-emergence, organophosphorus herbicide. Anilofos has moderate toxic potential in mammals[1].

  • CAS Number: 64249-01-0
  • MF: C13H19ClNO3PS2
  • MW: 367.85200
  • Catalog: Others
  • Density: 1.322 g/cm3
  • Boiling Point: 443.6ºC at 760 mmHg
  • Melting Point: 50-51ºC
  • Flash Point: >100 °C

Idarucizumab

Idarucizumab is a humanized monoclonal antibody fragment. Idarucizumab is first reversal agent for a direct oral anticoagulant (DOAC). Idarucizumab can specifically neutralize the effects of the oral direct thrombin inhibitor in order to restore hemostasis[1].

  • CAS Number: 1362509-93-0
  • MF:
  • MW:
  • Catalog: Cardiovascular Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-Ser(PO(NHPr)2)-OH

Fmoc-Ser(PO(NHPr)2)-OH is a serine derivative[1].

  • CAS Number: 216061-08-4
  • MF: C24H32N3O6P
  • MW: 489.50
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-L-Ser-Obzl

Fmoc-Ser-Obzl is a serine derivative[1].

  • CAS Number: 73724-46-6
  • MF: C25H23NO5
  • MW: 417.454
  • Catalog: Others
  • Density: 1.279±0.06 g/cm3
  • Boiling Point: 656.2±55.0 °C at 760 mmHg
  • Melting Point: 98-100 ºC
  • Flash Point: 350.7±31.5 °C

Iso-mogroside V

Isomogroside V is a sweetener, which extracted from Siraitia grosvenorii (Swingle).

  • CAS Number: 1126032-65-2
  • MF: C60H102O29
  • MW: 1287.434
  • Catalog: Others
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1,5-Dihydroxypentane-d10

1,5-Dihydroxypentane-d10 is the deuterium labeled 1,5-Dihydroxypentane[1].

  • CAS Number: 1219804-42-8
  • MF: C5H2D10O2
  • MW: 114.209
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 239.0±0.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 129.4±0.0 °C

Mca-KKEDVV-Abu-C

Mca-KKEDVV-Abu-C is a peptide. Mca-KKEDVV-Abu-C can be used for various biochemical researches.

  • CAS Number: 290836-22-5
  • MF: C50H76N10O17S
  • MW: 1121.26
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Eftansomatropin alfa

Eftansomatropin alfa is an antibody targeting the growth hormone receptor (GSH). Eftansomatropin alfa is a fusion protein of GH1 and IGHG4 Fc[1].

  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Phensuximide

Phensuximide is an orally active succinimide antiepileptic and anticonvulsant agent. Phensuximide inhibits cyclic AMP and cyclic GMP accumulation in depolarized brain tissue. Phensuximide can be used for the study of seizure and petit mal[1][3].

  • CAS Number: 86-34-0
  • MF: C11H11NO2
  • MW: 189.21100
  • Catalog: Others
  • Density: 1.1596 (rough estimate)
  • Boiling Point: 324.47°C (rough estimate)
  • Melting Point: 71-73°
  • Flash Point: N/A

LHRH (lamprey III) trifluoroacetate salt

LGnRH-III, lamprey, an isoform of GnRH isolated from the sea lamprey, is a weak GnRH agonist with antitumor activities[1][2].

  • CAS Number: 147859-97-0
  • MF: C59H74N18O14
  • MW: 1259.33
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

IEIK 13

IEIK 13 is a self-assembling peptide (SAP) sequence. IEIK 13 can be used for the research of cartilage tissue engineering[1]

  • CAS Number: 1426415-02-2
  • MF: C77H139N17O20
  • MW: 1623.03
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

diftalone

Diftalone (Aladione) is an anti-inflammatory agent. Diftalone can be used for research of inflammatory disease, such as rheumatoid arthritis[1].

  • CAS Number: 21626-89-1
  • MF: C16H12N2O2
  • MW: 264.27900
  • Catalog: Inflammation/Immunology
  • Density: 1.43g/cm3
  • Boiling Point: 462ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 221.2ºC

PAF-AN-1

PAF-AN-1 is a platelet activating factor receptor (PAF) antagonist.

  • CAS Number: 115621-84-6
  • MF: C28H28N2O3
  • MW: 440.53
  • Catalog: Cardiovascular Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Condurango glycoside C

Condurango glycoside C is isolated from the bark of Marsdenia eunduranog [1].

  • CAS Number: 11051-92-6
  • MF: C53H80O17
  • MW: 989.19
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

ML154

ML154 is a potent antagonist of NPSR. ML154 has the potential for the research of anxiety, addiction and food disorders[1].

  • CAS Number: 1345964-89-7
  • MF: C29H26BrN2PS
  • MW: 261.29600
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Polyquaternium-1

Polyquaternium-1 (Polidronium chloride) is a polycationic ophthalmic preservative. Polyquaternium-1 can inhibit growth of microbial contaminants in multi-dose bottles of topical medications[1].

  • CAS Number: 75345-27-6
  • MF: C22H48Cl3N3O6
  • MW: 810.21
  • Catalog: Infection
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-PALMITOYL(D31)-2-OLEOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE

16:0-18:1 PE-d31 is deuterium labeled 16:0-18:1 PE.

  • CAS Number: 326495-44-7
  • MF: C39H45D31NO8P
  • MW: 749.187
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 741.6±70.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 402.3±35.7 °C

Methyl N-[(benzyloxy)carbonyl]-D-serinate

Methyl ((benzyloxy)carbonyl)-D-serinate is a serine derivative[1].

  • CAS Number: 93204-36-5
  • MF: C12H15NO5
  • MW: 253.251
  • Catalog: Others
  • Density: 1.254g/cm3
  • Boiling Point: 442.6±45.0 °C at 760 mmHg
  • Melting Point: 41-43ºC(lit.)
  • Flash Point: 221.5±28.7 °C

asperlicin D

Asperlicin D is a asperlicin productionfrom Aspergillus alliaceus strain (ATCC 20656)[1].

  • CAS Number: 93413-07-1
  • MF: C25H18N4O2
  • MW: 406.43600
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

O-Methyl-O-(N-butylfluorescein)phosphate

O-Methyl-O-(N-butylfluorescein)phosphate is a fluorescent dye.

  • CAS Number: 887406-94-2
  • MF: C25H23O8P
  • MW: 482.41900
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Boc-beta-alanine

Boc-β-Ala-OH is an alanine derivative[1].

  • CAS Number: 3303-84-2
  • MF: C8H15NO4
  • MW: 189.209
  • Catalog: Others
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 320.9±25.0 °C at 760 mmHg
  • Melting Point: 76-78 °C
  • Flash Point: 147.9±23.2 °C

WZB 117

WZB117 is a glucose transporter 1 (Glut1) inhibitor, which downregulates glycolysis, induces cell-cycle arrest, and inhibits cancer cell growth in vitro and in vivo.

  • CAS Number: 1223397-11-2
  • MF: C20H13FO6
  • MW: 368.312
  • Catalog: Cancer
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 628.4±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 333.9±31.5 °C

D-JBD19

D-JBD19 is a non-permeable peptide[1]. D-JBD19 has neuroprotective effects[2].

  • CAS Number: 954134-42-0
  • MF: C99H164N32O28
  • MW: 2250.56
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

H-Ala-OtBu.HCl

H-Ala-OtBu.HCl is an alanine derivative[1].

  • CAS Number: 13404-22-3
  • MF: C7H16ClNO2
  • MW: 181.660
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 206.8ºC at 760 mmHg
  • Melting Point: 168-175 °C (dec.)
  • Flash Point: 78.9ºC

DABCYL-TNF-α-EDANS (-4 to +6) (human) trifluoroacetate salt

DABCYL-TNF-α-EDANS (-4 to +6) (human) is a FRET peptide substrate of tumor necrosis factor convertase (TACE)[1].

  • CAS Number: 396716-14-6
  • MF: C70H104N22O18S
  • MW: 1573.776
  • Catalog: Cancer
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

HOE-S 785026

HOE-S 785026 is a blue fluorescent dyes, which can be used as a cell dye for DNA.

  • CAS Number: 132869-83-1
  • MF: C25H24N6O
  • MW: 424.49800
  • Catalog: Dye Reagents
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

H-Gly-Gly-Met-OH

H-Gly-Gly-Met-OH is a biologically active peptide.

  • CAS Number: 17343-02-1
  • MF: C9H17N3O4S
  • MW: 263.31400
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

HSMO9

HSMO9 is a (+)-methamphetamine (METH)-like hapten that can be coupled to a carrier protein. HSMO9 can be used in vaccine development[1].

  • CAS Number: 1313762-77-4
  • MF: C18H30N2O2S
  • MW: 338.51
  • Catalog: Inflammation/Immunology
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

CD147 degrader 1

CD147 degrader 1 is a PROTAC targets CD147 with an DC50 value of 6.72 µM. CD147 degrader 1 inhibits cell proliferation, migration and invasion. CD147 degrader 1 decreases the expression of CD147, MMP9, and p-STAT3 protein. CD147 degrader 1 shows anti-cancer acyivity[1].

  • CAS Number: 2416740-37-7
  • MF: C38H42N4O11
  • MW: 730.76
  • Catalog: PROTAC
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Betamethasone Acetate

Betamethasone acetate is a glucocorticoid corticosteroid. Betamethasone acetate induces fetal lung maturation in preterm sheep[1].

  • CAS Number: 987-24-6
  • MF: C24H31FO6
  • MW: 434.498
  • Catalog: Inflammation/Immunology
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 579.4±50.0 °C at 760 mmHg
  • Melting Point: 200-220°C (dec.)
  • Flash Point: 304.2±30.1 °C