Chemsrc provides Others's classification. They are divided into Androgen Receptor, Aromatase, Estrogen Receptor/ERR, Progesterone Receptor, Thyroid Hormone Receptor, Others according to their Biological activity.


Anti-infection >
Arenavirus Bacterial CMV Enterovirus Filovirus Fungal HBV HCV HIV HSV Influenza Virus Parasite Reverse Transcriptase RSV SARS-CoV
Antibody-drug Conjugate >
ADC Cytotoxin ADC Linker Drug-Linker Conjugates for ADC PROTAC-linker Conjugate for PAC
Apoptosis >
Apoptosis Bcl-2 Family c-Myc Caspase DAPK Ferroptosis IAP MDM-2/p53 PKD RIP kinase Survivin Thymidylate Synthase TNF Receptor
Autophagy >
Autophagy LRRK2 ULK Mitophagy
Cell Cycle/DNA Damage >
Antifolate APC ATM/ATR Aurora Kinase Casein Kinase CDK Checkpoint Kinase (Chk) CRISPR/Cas9 Deubiquitinase DNA Alkylator/Crosslinker DNA-PK DNA/RNA Synthesis Eukaryotic Initiation Factor (eIF) G-quadruplex Haspin Kinase HDAC HSP IRE1 Kinesin LIM Kinase (LIMK) Microtubule/Tubulin Mps1 Nucleoside Antimetabolite/Analog p97 PAK PARP PERK Polo-like Kinase (PLK) PPAR RAD51 ROCK Sirtuin SRPK Telomerase TOPK Topoisomerase Wee1
Cytoskeleton >
Arp2/3 Complex Dynamin Gap Junction Protein Integrin Kinesin Microtubule/Tubulin Mps1 Myosin PAK
Epigenetics >
AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain HDAC Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MicroRNA PARP PKC Sirtuin Protein Arginine Deiminase
GPCR/G Protein >
5-HT Receptor Adenosine Receptor Adenylate Cyclase Adiponectin Receptor Adrenergic Receptor Angiotensin Receptor Bombesin Receptor Bradykinin Receptor Cannabinoid Receptor CaSR CCR CGRP Receptor Cholecystokinin Receptor CRFR CXCR Dopamine Receptor EBI2/GPR183 Endothelin Receptor GHSR Glucagon Receptor Glucocorticoid Receptor GNRH Receptor GPCR19 GPR109A GPR119 GPR120 GPR139 GPR40 GPR55 GPR84 Guanylate Cyclase Histamine Receptor Imidazoline Receptor Leukotriene Receptor LPL Receptor mAChR MCHR1 (GPR24) Melatonin Receptor mGluR Motilin Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor Opioid Receptor Orexin Receptor (OX Receptor) Oxytocin Receptor P2Y Receptor Prostaglandin Receptor Protease-Activated Receptor (PAR) Ras RGS Protein Sigma Receptor Somatostatin Receptor TSH Receptor Urotensin Receptor Vasopressin Receptor Melanocortin Receptor
Immunology/Inflammation >
Aryl Hydrocarbon Receptor CCR Complement System COX CXCR FLAP Histamine Receptor IFNAR Interleukin Related IRAK MyD88 NO Synthase NOD-like Receptor (NLR) PD-1/PD-L1 PGE synthase Salt-inducible Kinase (SIK) SPHK STING Thrombopoietin Receptor Toll-like Receptor (TLR) Arginase
JAK/STAT Signaling >
EGFR JAK Pim STAT
MAPK/ERK Pathway >
ERK JNK KLF MAP3K MAP4K MAPKAPK2 (MK2) MEK Mixed Lineage Kinase MNK p38 MAPK Raf Ribosomal S6 Kinase (RSK)
Membrane Transporter/Ion Channel >
ATP Synthase BCRP Calcium Channel CFTR Chloride Channel CRAC Channel CRM1 EAAT2 GABA Receptor GlyT HCN Channel iGluR Monoamine Transporter Monocarboxylate Transporter Na+/Ca2+ Exchanger Na+/HCO3- Cotransporter Na+/K+ ATPase nAChR NKCC P-glycoprotein P2X Receptor Potassium Channel Proton Pump SGLT Sodium Channel TRP Channel URAT1
Metabolic Enzyme/Protease >
15-PGDH 5 alpha Reductase 5-Lipoxygenase Acetyl-CoA Carboxylase Acyltransferase Adenosine Deaminase Adenosine Kinase Aldehyde Dehydrogenase (ALDH) Aldose Reductase Aminopeptidase Angiotensin-converting Enzyme (ACE) ATGL ATP Citrate Lyase Carbonic Anhydrase Carboxypeptidase Cathepsin CETP COMT Cytochrome P450 Dipeptidyl Peptidase Dopamine β-hydroxylase E1/E2/E3 Enzyme Elastase Enolase FAAH FABP Factor Xa Farnesyl Transferase Fatty Acid Synthase (FAS) FXR Glucokinase GSNOR Gutathione S-transferase HCV Protease Hexokinase HIF/HIF Prolyl-Hydroxylase HIV Integrase HIV Protease HMG-CoA Reductase (HMGCR) HSP Indoleamine 2,3-Dioxygenase (IDO) Isocitrate Dehydrogenase (IDH) Lactate Dehydrogenase LXR MAGL Mineralocorticoid Receptor Mitochondrial Metabolism MMP Nampt NEDD8-activating Enzyme Neprilysin PAI-1 PDHK PGC-1α Phosphatase Phosphodiesterase (PDE) Phospholipase Procollagen C Proteinase Proteasome Pyruvate Kinase RAR/RXR Renin ROR Ser/Thr Protease SGK Stearoyl-CoA Desaturase (SCD) Thrombin Tryptophan Hydroxylase Tyrosinase Xanthine Oxidase
Neuronal Signaling >
5-HT Receptor AChE Adenosine Kinase Amyloid-β Beta-secretase CaMK CGRP Receptor COMT Dopamine Receptor Dopamine Transporter FAAH GABA Receptor GlyT iGluR Imidazoline Receptor mAChR Melatonin Receptor Monoamine Oxidase nAChR Neurokinin Receptor Opioid Receptor Serotonin Transporter γ-secretase
NF-κB >
NF-κB IKK Keap1-Nrf2 MALT1
PI3K/Akt/mTOR >
Akt AMPK ATM/ATR DNA-PK GSK-3 MELK mTOR PDK-1 PI3K PI4K PIKfyve PTEN
PROTAC >
PROTAC E3 Ligase Ligand-Linker Conjugate Ligand for E3 Ligase PROTAC Linker PROTAC-linker Conjugate for PAC
Protein Tyrosine Kinase/RTK >
Ack1 ALK Bcr-Abl BMX Kinase Btk c-Fms c-Kit c-Met/HGFR Discoidin Domain Receptor DYRK EGFR Ephrin Receptor FAK FGFR FLT3 IGF-1R Insulin Receptor IRAK Itk PDGFR PKA Pyk2 ROS Src Syk TAM Receptor Trk Receptor VEGFR
Stem Cell/Wnt >
Casein Kinase ERK Gli GSK-3 Hedgehog Hippo (MST) JAK Notch Oct3/4 PKA Porcupine ROCK sFRP-1 Smo STAT TGF-beta/Smad Wnt YAP β-catenin γ-secretase
TGF-beta/Smad >
TGF-beta/Smad PKC ROCK TGF-β Receptor
Vitamin D Related >
VD/VDR
Others >
Androgen Receptor Aromatase Estrogen Receptor/ERR Progesterone Receptor Thyroid Hormone Receptor Others

TAT-amide

TAT-amide is a cell penetrating peptide. Cell-penetrating peptides (CPPs) are short amino acid sequences able to enter different cells[1][2].

  • CAS Number: 697226-52-1
  • MF: C64H119N33O13
  • MW: 1558.84
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Trofinetide

Trofinetide, a synthetic analogue of the endogenous N-terminus tripeptide, Glycine-Proline-Glutamate (GPE), has been shown to be neuroprotective in animal models of brain injury.

  • CAS Number: 853400-76-7
  • MF: C13H21N3O6
  • MW: 315.322
  • Catalog: Neurological Disease
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 655.4±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 350.2±31.5 °C

INH6

INH6 is a potent Nek2/Hec1 inhibitor; inhibits the growth of HeLa cells with an IC50 of 2.4 μM.

  • CAS Number: 1001753-24-7
  • MF: C19H18N2OS
  • MW: 322.424
  • Catalog: Cancer
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Boc-Glu(OBzl)-Osu

Boc-Glu(OBzl)-OSu can be used for the solid-phase peptide synthesis containing glutamate benzyl ester residues.

  • CAS Number: 32886-40-1
  • MF: C21H26N2O8
  • MW: 434.440
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

1-bromooctane-1,1-d2

1-Bromooctane-1,1-d2 is the deuterium labeled 1-Bromooctane[1].

  • CAS Number: 86423-34-9
  • MF: C8H15BrD2
  • MW: 195.13700
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

10-(3-Sulfopropyl)acridinium betaine

10-(3-Sulfopropyl)acridinium Betaine is a fluorescent dye with high durability (>3 months)[1].

  • CAS Number: 83907-41-9
  • MF: C16H15NO3S
  • MW: 301.36000
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 280-290ºC (dec.)
  • Flash Point: N/A

Protoescigenin

Protoescigenin is the main aglycone of horse chestnut saponin mixture known as escin. Protoescigenin is selected as substrate for exploratory chemistry towards selective protection, followed by propargyl ether formation and subsequent condensation with azido-monosaccharides, to obtain novel triazole linked conjugates of the triterpene[1].

  • CAS Number: 20853-07-0
  • MF: C30H50O6
  • MW: 506.714
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 634.5±55.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 262.0±26.1 °C

4'-Demethyldehydropodophyllotoxin

4'-Demethyldehydropodophyllotoxin is an aryltetralin lignan that can be isolated from leaves of Podophyllum hexandrum. 4'-Demethyldehydropodophyllotoxin exhibits some cytotoxic and antitumour activity[1].

  • CAS Number: 117669-31-5
  • MF: C21H16O8
  • MW: 396.35
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fmoc-Lys-OAll.HCl

Fmoc-Lys-OAll.HCl is a lysine derivative[1].

  • CAS Number: 815619-80-8
  • MF: C24H29ClN2O4
  • MW: 444.951
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Boc-L-Leu-NMe(OMe)

(S)-N-Methyl-N-methoxy-2-(tert-butoxycarbonylamino)-4-methylpentanamide is a leucine derivative[1].

  • CAS Number: 87694-50-6
  • MF: C13H26N2O4
  • MW: 274.357
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 418.9±30.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 207.1±24.6 °C

Ds-HAPP

Ds-HAPP is an anthrancenyl and dansyl fluorophore ligand.

  • CAS Number: 330163-26-3
  • MF: C22H35N5O2S
  • MW: 433.61
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Fentiazac

Fentiazac, alkanoic acid derivative, is an orally active non-steroidal anti-inflammatory agent, with analgesic, antipyretic and platelet anti-aggregation activity. Fentiazac can be used to research inflammatory diseases such as rheumatoid arthritis, osteoarthritis and tendinitis[1][2][3].

  • CAS Number: 18046-21-4
  • MF: C17H12ClNO2S
  • MW: 329.80100
  • Catalog: Inflammation/Immunology
  • Density: 1.362g/cm3
  • Boiling Point: 556.2ºC at 760mmHg
  • Melting Point: 162ºC
  • Flash Point: 290.2ºC

GDC-0927 R-form

GDC-0927 (SRN-927, RG-6047) is a potent, orally bioavailable, selective estrogen receptor degrader (SERD) for treatment of metastatic hormone receptor-positive/HER2-negative breast cancer.

  • CAS Number: 1642297-53-7
  • MF: C28H28FNO4
  • MW: 461.533
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

9-Nitro(2H9)anthracene

9-Nitroanthracene-d9 is the deuterium labeled 9-Nitroanthracene[1].

  • CAS Number: 220381-38-4
  • MF: C14D9NO2
  • MW: 232.282
  • Catalog: Others
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 402.9±14.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 200.4±12.9 °C

denatonium benzoate

Denatonium is the most bitter chemical compound known,used as aversive agents (bitterants) to prevent inappropriate ingestion. Denatonium is used in denatured alcohol, antifreeze, nail biting preventions, respirator mask fit-testing, animal repellents, liquid soaps, and shampoos.

  • CAS Number: 3734-33-6
  • MF: C28H34N2O3
  • MW: 446.581
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: 164-168 °C(lit.)
  • Flash Point: N/A

glycine tert-butyl ester dibenzenesulfimide salt

Glycine tert-butyl ester dibenzenesulfonimide salt is a Glycine (HY-Y0966) derivative[1].

  • CAS Number: 77284-30-1
  • MF: C18H24N2O6S2
  • MW: 428.52300
  • Catalog: Others
  • Density: N/A
  • Boiling Point: 566.6ºC at 760 mmHg
  • Melting Point: 154-157ºC (dec.)
  • Flash Point: 296.4ºC

8,8''-Bibaicalein

8,8''-Bibaicalein is a natural product that can be found in baicalensis[1].

  • CAS Number: 135309-02-3
  • MF: C30H18O10
  • MW: 538.458
  • Catalog: Others
  • Density: 1.7±0.1 g/cm3
  • Boiling Point: 928.2±65.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 314.4±27.8 °C

7-beta-Hydroxylathyrol

7beta-Hydroxylathyrol is a natural product.

  • CAS Number: 34208-98-5
  • MF: C20H30O5
  • MW: 350.449
  • Catalog: Others
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 548.6±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 299.7±26.6 °C

Antiproliferative agent-41

Antiproliferative agent-41 (compound 14) is a antiproliferative agent indanorine[1].

  • CAS Number: 225652-93-7
  • MF: C20H20O4
  • MW: 324.37
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

HPA-12

HPA-12 is an intracellular ceramide transport protein inhibitor[1].

  • CAS Number: 383418-30-2
  • MF: C22H37NO3
  • MW: 363.54
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Exherin (trifluoroacetate)

Exherin trifluoroacetate is an N-cadherin antagonist, which inhibits N-cadherin mediated cell adhesion.

  • CAS Number: 1135237-88-5
  • MF: C24H35F3N8O8S2
  • MW: 684.70900
  • Catalog: Cancer
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Glimepiride-d4(phenylethyl-α,α,β,β-d4)(cis/trans)

Glimepiride-d4(phenylethyl-α,α,β,β-d4)(cis/trans) is the deuterium labeled [1].

  • CAS Number: 2699607-96-8
  • MF: C24H30D4N4O5S
  • MW: 494.64
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

PolQi2

PolQi2 inhibits the helicase activity of Polθ. PolQi2 improves the precision of gene editing at various loci and in different cell lines[1].

  • CAS Number: 2565638-16-4
  • MF: C21H16ClN5O3S
  • MW: 453.90
  • Catalog: Others
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Lauryl aldehyde

Dodecanal is composition of essential oil that can be found in Coriandrum sativum L.[1]

  • CAS Number: 112-54-9
  • MF: C12H24O
  • MW: 184.318
  • Catalog: Others
  • Density: 0.8±0.1 g/cm3
  • Boiling Point: 242.2±3.0 °C at 760 mmHg
  • Melting Point: 12 °C
  • Flash Point: 102.0±6.0 °C

CP 154526

CP 154526, a non peptidic corticotropin releasing factor receptor antagonist attenuates fever and exhibits anxiolytic-like activity[1].

  • CAS Number: 157286-86-7
  • MF: C23H32N4
  • MW: 364.52700
  • Catalog: Neurological Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Estradiol dipropionate

Estradiol dipropionate is a combined estrogen-progesterone, acts as an estrogen and progesterone agonist[1].

  • CAS Number: 113-38-2
  • MF: C24H32O4
  • MW: 384.50800
  • Catalog: Endocrinology
  • Density: 1.14g/cm3
  • Boiling Point: 487.8ºC at 760mmHg
  • Melting Point: 104-106℃ (ethanol )
  • Flash Point: 238.5ºC

Pipebuzone

Pipebuzone (LD 4644) is an anti-inflammatory, antipyretic and analgesic agent. Pipebuzone plays an important raol in rheumatic diseases[1].

  • CAS Number: 27315-91-9
  • MF: C25H32N4O2
  • MW: 420.54700
  • Catalog: Inflammation/Immunology
  • Density: 1.157g/cm3
  • Boiling Point: 530.6ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 208ºC

Clinopodiside A

Clinopodiside A, a triterpenoid saponin, is isolated from Clinopodium polycephalum which is a popular Chinese traditional medicinal herb[1][2].

  • CAS Number: 142809-89-0
  • MF: C48H78O19
  • MW: 959.12200
  • Catalog: Others
  • Density: 1.46g/cm3
  • Boiling Point: 1073.2ºC at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 602.9ºC

Pterodondiol

Pterodondiol is a gandular trichome metabolite on the leaves of Laggera pterodonta[1].

  • CAS Number: 60132-35-6
  • MF: C15H28O2
  • MW: 240.38
  • Catalog: Others
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 317.3±10.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 137.3±13.6 °C

APJ receptor agonist 5

APJ receptor agonist 5 (compound 3) is a potent and orally active agonist of apelin receptor (APJ) with an EC50 of 0.4 nM. APJ receptor agonist 5 displays excellent pharmacokinetic profiles in the rodent heart failure (HF) model. APJ receptor agonist 5 also shows an acceptable safety profile in preclinical toxicology studies. APJ receptor agonist 5 leads to improved cardiac function and can be used for researching the HF disease[1].

  • CAS Number: 2135514-20-2
  • MF: C26H29N3O6
  • MW: 479.52
  • Catalog: Cardiovascular Disease
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A