CB1R antagonist 1
Modify Date: 2024-04-06 16:37:24
CB1R antagonist 1 structure
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Common Name | CB1R antagonist 1 | ||
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| CAS Number | 334668-69-8 | Molecular Weight | 404.45 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C18H23F3N2O3S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of CB1R antagonist 1CB1R Allosteric modulator 5, a novel1-sulfonyl-4-acylpiperazines as selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC50 value of 4.2 μM and EC50 value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity[1]. |
| Name | CB1R antagonist 1 |
|---|
| Description | CB1R Allosteric modulator 5, a novel1-sulfonyl-4-acylpiperazines as selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC50 value of 4.2 μM and EC50 value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity[1]. |
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| Related Catalog | |
| Target |
hCB1-R:4.2 μM (IC50) hCB1-R:10 μM (EC50) |
| In Vitro | CB1R Allosteric modulator 5 has cannabinoid-1 receptor (CB1R) activity with an IC50value of 4.2 μM and EC50 value of ＞10 μM[1]. |
| References |
| Molecular Formula | C18H23F3N2O3S |
|---|---|
| Molecular Weight | 404.45 |