ERα antagonist 1

Modify Date: 2025-08-25 22:03:13

ERα antagonist 1 Structure
ERα antagonist 1 structure
Common Name ERα antagonist 1
CAS Number 2762423-09-4 Molecular Weight 568.68
Density N/A Boiling Point N/A
Molecular Formula C33H32N2O5S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of ERα antagonist 1


ERα antagonist 1 (Compound 19d) is a potent, selective, covalent estrogen receptor α (ERα) antagonist. ERα antagonist 1 induces apoptosis and cell cycle G0/G1 phase arrest in MCF-7 cells[1].

 Names

Name ERα antagonist 1

 ERα antagonist 1 Biological Activity

Description ERα antagonist 1 (Compound 19d) is a potent, selective, covalent estrogen receptor α (ERα) antagonist. ERα antagonist 1 induces apoptosis and cell cycle G0/G1 phase arrest in MCF-7 cells[1].
Related Catalog
Target

ERα

References

[1]. Bai C, et al. Benzothiophene derivatives as selective estrogen receptor covalent antagonists: Design, synthesis and anti-ERα activities. Bioorg Med Chem. 2021 Oct 1;47:116395.

 Chemical & Physical Properties

Molecular Formula C33H32N2O5S
Molecular Weight 568.68
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