ERα antagonist 1

Modify Date: 2024-01-08 12:01:12

ERα antagonist 1 structure	Common Name	ERα antagonist 1
	CAS Number	2762423-09-4	Molecular Weight	568.68
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₃₃H₃₂N₂O₅S	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of ERα antagonist 1

ERα antagonist 1 (Compound 19d) is a potent, selective, covalent estrogen receptor α (ERα) antagonist. ERα antagonist 1 induces apoptosis and cell cycle G0/G1 phase arrest in MCF-7 cells[1].

Name	ERα antagonist 1

Description	ERα antagonist 1 (Compound 19d) is a potent, selective, covalent estrogen receptor α (ERα) antagonist. ERα antagonist 1 induces apoptosis and cell cycle G0/G1 phase arrest in MCF-7 cells[1].
Related Catalog	Signaling Pathways >> Others >> Estrogen Receptor/ERR Signaling Pathways >> Apoptosis >> Apoptosis Research Areas >> Cancer
Target	ERα
References	[1]. Bai C, et al. Benzothiophene derivatives as selective estrogen receptor covalent antagonists: Design, synthesis and anti-ERα activities. Bioorg Med Chem. 2021 Oct 1;47:116395.

Molecular Formula	C₃₃H₃₂N₂O₅S
Molecular Weight	568.68