334668-69-8
334668-69-8 structure
- Name: CB1R antagonist 1
- Chemical Name: CB1R antagonist 1
- CAS Number: 334668-69-8
- Molecular Formula: C18H23F3N2O3S
- Molecular Weight: 404.45
- Catalog: Signaling Pathways GPCR/G Protein Cannabinoid Receptor
- Create Date: 2022-09-16 09:37:56
- Modify Date: 2024-04-06 16:37:24
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CB1R Allosteric modulator 5, a novel1-sulfonyl-4-acylpiperazines as selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC50 value of 4.2 μM and EC50 value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity[1].
| Name | CB1R antagonist 1 |
|---|
| Description | CB1R Allosteric modulator 5, a novel1-sulfonyl-4-acylpiperazines as selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC50 value of 4.2 μM and EC50 value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity[1]. |
|---|---|
| Related Catalog | |
| Target |
hCB1-R:4.2 μM (IC50) hCB1-R:10 μM (EC50) |
| In Vitro | CB1R Allosteric modulator 5 has cannabinoid-1 receptor (CB1R) activity with an IC50value of 4.2 μM and EC50 value of ＞10 μM[1]. |
| References |
| Molecular Formula | C18H23F3N2O3S |
|---|---|
| Molecular Weight | 404.45 |