CCR2 antagonist 1

Modify Date: 2024-01-11 20:37:32

CCR2 antagonist 1 structure	Common Name	CCR2 antagonist 1
	CAS Number	1683534-96-4	Molecular Weight	549.47
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₈H₃₂BrF₃N₂O	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of CCR2 antagonist 1

CCR2 antagonist 1 is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM.

Name	CCR2 antagonist 1

Description	CCR2 antagonist 1 is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> CCR Signaling Pathways >> Immunology/Inflammation >> CCR Research Areas >> Others
Target	CCR2:2.4 nM (Ki)
In Vitro	The combination of SAR and SKR in the hit-to-lead process results in the discovery of a new higheaffinity and longeresidenceetime CCR2 antagonist (CCR2 antagonist 1 (compound 15a), Ki=2.4 nM; RT=714 min)[1].
References	[1]. Vilums M, et al. When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists. Eur J Med Chem. 2015 Mar 26;93:121-34.

Molecular Formula	C₂₈H₃₂BrF₃N₂O
Molecular Weight	549.47

DC Chemicals Limited
China
Product Name: CCR2 antagonist 1
Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/1g
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

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