1683534-96-4
1683534-96-4 structure
- Name: CCR2 antagonist 1
- Chemical Name: CCR2 antagonist 1
- CAS Number: 1683534-96-4
- Molecular Formula: C28H32BrF3N2O
- Molecular Weight: 549.47
- Catalog: Signaling Pathways GPCR/G Protein CCR
- Create Date: 2019-02-08 09:13:50
- Modify Date: 2025-08-27 02:01:08
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CCR2 antagonist 1 is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM.
| Name | CCR2 antagonist 1 |
|---|
| Description | CCR2 antagonist 1 is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM. |
|---|---|
| Related Catalog | |
| Target |
CCR2:2.4 nM (Ki) |
| In Vitro | The combination of SAR and SKR in the hit-to-lead process results in the discovery of a new higheaffinity and longeresidenceetime CCR2 antagonist (CCR2 antagonist 1 (compound 15a), Ki=2.4 nM; RT=714 min)[1]. |
| References |
| Molecular Formula | C28H32BrF3N2O |
|---|---|
| Molecular Weight | 549.47 |