hGPR91 antagonist 1

Modify Date: 2025-08-20 10:32:55

hGPR91 antagonist 1 structure	Common Name	hGPR91 antagonist 1
	CAS Number	1314796-00-3	Molecular Weight	529.53
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₃₁H₂₃F₄N₃O	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of hGPR91 antagonist 1

HGPR91 antagonist 1 is a potent and selective small molecule hGPR91 antagonist with an IC50 of 7 μM[1].

Name	hGPR91 antagonist 1

Description	HGPR91 antagonist 1 is a potent and selective small molecule hGPR91 antagonist with an IC50 of 7 μM[1].
Related Catalog	Research Areas >> Others Signaling Pathways >> Others >> Others
Target	IC50: 7 μM (HGPR91)[1]
In Vivo	HGPR91 antagonist 1 leads to 59, 76% inhibition of ΔMAP at 2, 4 hours and has shown rat plasma protein binding 99%. HGPR91 antagonist 1 has engaged the target under the in vivo condition. HGPR91 antagonist 1 has clearance (CL) of 0.2 nmol/min/mg of RLM[1]. Animal Model: Wistar rats[1] Dosage: 100 mg/kg Administration: I.p.; 2 and 4 hours Result: Led to 59 and 76% inhibition of ΔMAP at 2 and 4 hours.
References	[1]. Bhuniya D, et al. Discovery of a potent and selective small molecule hGPR91 antagonist. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3596-602.

Molecular Formula	C₃₁H₂₃F₄N₃O
Molecular Weight	529.53

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