Cavα2δ1&NET-IN-3

Modify Date: 2024-01-30 11:28:10

Cavα2δ1&NET-IN-3 Structure
Cavα2δ1&NET-IN-3 structure
Common Name Cavα2δ1&NET-IN-3
CAS Number 2143584-82-9 Molecular Weight 466.60
Density N/A Boiling Point N/A
Molecular Formula C24H30N6O2S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Cavα2δ1&NET-IN-3


Cavα2δ1&NET-IN-3 (example 216) is an inhibitor of the subunit α2δ of voltage-gated calcium channels (VGCC) and noradrenaline transporter (NET). Cavα2δ1&NET-IN-3 has Kis of 100-500 nM for human α2δ-1 subunit of Cav2.2 calcium channel and NET, respectively[1].

 Names

Name Cavα2δ1&NET-IN-3

 Cavα2δ1&NET-IN-3 Biological Activity

Description Cavα2δ1&NET-IN-3 (example 216) is an inhibitor of the subunit α2δ of voltage-gated calcium channels (VGCC) and noradrenaline transporter (NET). Cavα2δ1&NET-IN-3 has Kis of 100-500 nM for human α2δ-1 subunit of Cav2.2 calcium channel and NET, respectively[1].
Related Catalog
Target

Calcium Channel

References

[1]. subunit α2δ of voltage-gated calcium channels (VGCC) and noradrenaline transporter (NET). Cavα2δ1&NET-IN-3 has kis of 100-500 nM for human α2δ-1 subunit of Cav2.2

 Chemical & Physical Properties

Molecular Formula C24H30N6O2S
Molecular Weight 466.60