CETP-IN-3

Modify Date: 2024-01-09 15:51:24

CETP-IN-3 Structure
CETP-IN-3 structure
Common Name CETP-IN-3
CAS Number 939391-31-8 Molecular Weight 704.50
Density N/A Boiling Point N/A
Molecular Formula C30H24F12N2O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CETP-IN-3


CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP. CETP-IN-3 for the CETP inhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) with IC50s of 0.002 μM and 0.06 μM, respectively[1].

 Names

Name CETP-IN-3

 CETP-IN-3 Biological Activity

Description CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP. CETP-IN-3 for the CETP inhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) with IC50s of 0.002 μM and 0.06 μM, respectively[1].
Related Catalog
References

[1]. Finlay HJ, et al. Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor. ACS Med Chem Lett. 2019 May 6; 10(6):911-916.

 Chemical & Physical Properties

Molecular Formula C30H24F12N2O4
Molecular Weight 704.50