PNU 282987
Modify Date: 2025-09-29 12:59:28
PNU 282987 structure
|
Common Name | PNU 282987 | ||
|---|---|---|---|---|
| CAS Number | 711085-63-1 | Molecular Weight | 264.75 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C14H17ClN2O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PNU 282987PNU-282987 (free base) (Compound C7) is a potent α7 nicotinic acetylcholine receptor (nAChR) agonist with an EC50 of 154 nM. PNU-282987 (free base) is also a functional antagonist of the 5-HT3 receptor with an IC50 of 4541 nM[1]. |
| Name | Benzamide, N-(3R)-1-azabicyclo[2.2.2]oct-3-yl-4-chloro- |
|---|---|
| Synonym | More Synonyms |
| Description | PNU-282987 (free base) (Compound C7) is a potent α7 nicotinic acetylcholine receptor (nAChR) agonist with an EC50 of 154 nM. PNU-282987 (free base) is also a functional antagonist of the 5-HT3 receptor with an IC50 of 4541 nM[1]. |
|---|---|
| Related Catalog | |
| Target |
5-HT3 Receptor |
| References |
| Molecular Formula | C14H17ClN2O |
|---|---|
| Molecular Weight | 264.75 |
| Hazard Codes | Xi |
|---|
| MFCD08703110 |