KTX-497 structure
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Common Name | KTX-497 | ||
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CAS Number | 2432993-46-7 | Molecular Weight | 854.92 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C45H49F3N8O6 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of KTX-497KTX-497 is an orally active IRAK4 degrader with a DC50 value of 3 nM. KTX-497 can be used for the research of oncology[1]. |
Name | KTX-497 |
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Description | KTX-497 is an orally active IRAK4 degrader with a DC50 value of 3 nM. KTX-497 can be used for the research of oncology[1]. |
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Related Catalog | |
Target |
IRAK4:3 nM (DC50) |
In Vitro | KTX-497 has activity for IRAK4 with a DC50 value of 3 nM[1]. |
In Vivo | KTX-497 (oral; 10 mg/kg) impacts oral absorption[1]. Animal Model: Rat[1] Dosage: 10 mg/kg Administration: Oral Result: Rat PO PK (10 mg/kg) KTX-497 %F 17 AUC(μM*hr) 1.4 |
References |
Molecular Formula | C45H49F3N8O6 |
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Molecular Weight | 854.92 |