5-溴-2-甲氧基吡啶
5-溴-2-甲氧基吡啶结构式
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常用名 | 5-溴-2-甲氧基吡啶 | 英文名 | 2-Methoxy-5-Bromopyridine |
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| CAS号 | 13472-85-0 | 分子量 | 188.02 | |
| 密度 | 1.5±0.1 g/cm3 | 沸点 | 197.0±20.0 °C at 760 mmHg | |
| 分子式 | C6H6BrNO | 熔点 | 80ºC (12 mmHg) | |
| MSDS | 中文版 美版 | 闪点 | 72.9±21.8 °C | |
| 符号 |
GHS07 |
信号词 | Warning |
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An efficient synthesis of an alphavbeta3 antagonist.
J. Org. Chem. 69 , 1959-1966, (2004) A practical preparation of an alpha(v)beta(3) antagonist is reported. The antagonist consists of three key components, a tetrahydronaphthyridine moiety, a beta-alanine moiety, and a central imidazolidone moiety. The tetrahydronaphthyridine component was prepa... |
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Non-peptide alpha v beta 3 antagonists. Part 7: 3-Substituted tetrahydro-naphthyridine derivatives.
Bioorg. Med. Chem. Lett. 14 , 1049, (2004) A series of 3-substituted tetrahydro-[1,8]naphthyridine containing alpha(v)beta(3) antagonists was prepared. A comparison of their in vitro IC(50) values to the electron properties of the 3-substituents revealed a good linear Hammett correlation (rho=-1.96, R... |
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Tetrahedron Asymmetry 14 , 3469, (2003)
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The 1,3-Diaminobenzene-Derived Aminophosphine Palladium Pincer Complex {C6H3[NHP(piperidinyl)2]2Pd(Cl)}-A Highly Active Suzuki-Miyaura Catalyst with Excellent Functional Group Tolerance. Bolliger JL and Frech CM.
Adv. Synth. Catal. 352(6) , 1075-1080, (2010)
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Functionalized pyridylboronic acids and their Suzuki cross-coupling reactions to yield novel heteroarylpyridines Parry PR, et al.
J. Org. Chem. 67(21) , 7541-7543, (2002)
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A scaleable synthesis of methyl 3-amino-5-(4-fluorobenzyl)-2-pyridinecarboxylate. Organic Process Research & Development 11.5 (2007): 899-902 Boros EE, et al. Org. Process Res. Dev. 11(5) , 899-902, (2007)
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Synthesis and biological evaluation of 1-(benzenesulfonamido)-2-[5-(N-hydroxypyridin-2 (1H)-one)] acetylene regioisomers: A novel class of 5-lipoxygenase inhibitors. Chowdhury MA, et al.
Bioorg. Med. Chem. Lett. 18(14) , 4195-4198, (2008)
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Negishi Cross-Coupling Reactions Catalyzed by an Aminophosphine-Based Nickel System: A Reliable and General Applicable Reaction Protocol for the High-Yielding Synthesis of Biaryls. Gerber R and Frech CM.
Chemistry 17(42) , 11893-11904, (2011)
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