A1AR antagonist 2

Modify Date: 2024-01-08 15:40:08

A1AR antagonist 2 Structure
A1AR antagonist 2 structure
Common Name A1AR antagonist 2
CAS Number 1441961-74-5 Molecular Weight 288.30
Density N/A Boiling Point N/A
Molecular Formula C17H12N4O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of A1AR antagonist 2


A1AR antagonist 2 (compound 18h) is a potent A1 adenosine receptor (AR) antagonist with Kis of 1.49, 10.2, and 50.1 nM for hA1, hA2A and hA2B, respectively[1].

 Names

Name A1AR antagonist 2

 A1AR antagonist 2 Biological Activity

Description A1AR antagonist 2 (compound 18h) is a potent A1 adenosine receptor (AR) antagonist with Kis of 1.49, 10.2, and 50.1 nM for hA1, hA2A and hA2B, respectively[1].
Related Catalog
References

[1]. Val C, et al. Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1 Antagonists. J Med Chem. 2022;65(3):2091-2106.

 Chemical & Physical Properties

Molecular Formula C17H12N4O
Molecular Weight 288.30