A1AR antagonist 5

Modify Date: 2025-08-22 22:16:45

A1AR antagonist 5 Structure
A1AR antagonist 5 structure
Common Name A1AR antagonist 5
CAS Number 1030509-01-3 Molecular Weight 326.78
Density N/A Boiling Point N/A
Molecular Formula C17H15ClN4O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of A1AR antagonist 5


A1AR antagonist 5 (compound 20) is a potent and selective A1AR (A1 adenosine receptor) antagonist, with a pIC50 of 5.83 and a pKi of 6.11[1].

 Names

Name A1AR antagonist 5

 A1AR antagonist 5 Biological Activity

Description A1AR antagonist 5 (compound 20) is a potent and selective A1AR (A1 adenosine receptor) antagonist, with a pIC50 of 5.83 and a pKi of 6.11[1].
Related Catalog
Target

hA1AR:6.11 (pKi)

hA2AAR:<4 (pKi)

References

[1]. Wei Y, et al. Identification of new potent A1 adenosine receptor antagonists using a multistage virtual screening approach. Eur J Med Chem. 2020 Feb 1;187:111936.

 Chemical & Physical Properties

Molecular Formula C17H15ClN4O
Molecular Weight 326.78
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.