2413257-73-3

2413257-73-3 structure

Name: A1AR antagonist 3
Chemical Name: A1AR antagonist 3
CAS Number: 2413257-73-3
Molecular Formula: C₂₅H₂₀N₂O₃S
Molecular Weight: 428.50
Catalog: Signaling Pathways GPCR/G Protein Adenosine Receptor
Create Date: 2022-08-30 17:19:36
Modify Date: 2025-08-25 17:53:42
A1AR antagonist 3 (compound 13) is a selective adenosine 1 (A1) receptor antagonist with Kis of 9.69 nM and 0.529 nM for human A1 and rat A1, respectively. A1AR antagonist 3 can be used for researching neurological diseases[1].

Name	A1AR antagonist 3

Description	A1AR antagonist 3 (compound 13) is a selective adenosine 1 (A1) receptor antagonist with Kis of 9.69 nM and 0.529 nM for human A1 and rat A1, respectively. A1AR antagonist 3 can be used for researching neurological diseases[1].
Related Catalog	Research Areas >> Neurological Disease Signaling Pathways >> GPCR/G Protein >> Adenosine Receptor
Target	human A1:9.69 nM (Ki) rat A1:0.529 nM (Ki)
References	[1]. Abdelrahman A, et al. Substituted 4-phenylthiazoles: Development of potent and selective A1, A3 and dual A1/A3 adenosine receptor antagonists. Eur J Med Chem. 2020;186:111879.

Molecular Formula	C₂₅H₂₀N₂O₃S
Molecular Weight	428.50