G Protein Antagonist
Modify Date: 2025-08-21 19:01:30
G Protein Antagonist structure
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Common Name | G Protein Antagonist | ||
|---|---|---|---|---|
| CAS Number | 143675-79-0 | Molecular Weight | 1093.26000 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C57H64N12O9S | Melting Point | N/A | |
| MSDS | Chinese USA | Flash Point | N/A | |
Use of G Protein AntagonistG-Protein antagonist peptide is the substance P-related peptide that inhibits binding of G proteins to their receptors. G-Protein antagonist peptide competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors. |
| Name | G-Protein antagonist peptide |
|---|---|
| Synonym | More Synonyms |
| Description | G-Protein antagonist peptide is the substance P-related peptide that inhibits binding of G proteins to their receptors. G-Protein antagonist peptide competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors. |
|---|---|
| Related Catalog |
| Molecular Formula | C57H64N12O9S |
|---|---|
| Molecular Weight | 1093.26000 |
| Exact Mass | 1092.46000 |
| PSA | 362.55000 |
| LogP | 6.16720 |
| InChIKey | WSYRBHQWMXTCHQ-SFIKJRKMSA-N |
| SMILES | CSCCC(NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C(Cc1ccccc1)NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C(CCC(N)=O)NC(=O)C1CCC(=O)N1)C(N)=O |
| Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
|---|---|
| Safety Phrases | 22-24/25 |
| RIDADR | NONH for all modes of transport |
| WGK Germany | 3 |
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G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding.
J. Biol. Chem. 267 , 16237, (1992) A substance P (SP) analog, [D-Pro4,D-Trp7,9,10] SP4-11, is known to inhibit the actions of various structurally unrelated messenger molecules as well as SP. Our studies on the effects of this peptide ... |
| PYR-GLN-D-TRP-PHE-D-TRP-D-TRP-MET-NH2 |
| pglu-gln-d-trp-phe-d-trp-d-trp-met-nh2 |
| G PROTEIN ANTAGONIST |
| PROTEIN G ANTAGONIST 2 |
| GP ANTAGONIST-2 |
| pGlu-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH2 |
| [pGlu5,D-Trp7,9,10]-Substance P Fragment 5-11 |
| G-PROTEIN ANTAGONIST-2 |