G Protein Antagonist

Modify Date: 2024-01-02 19:49:07

G Protein Antagonist structure	Common Name	G Protein Antagonist
	CAS Number	143675-79-0	Molecular Weight	1093.26000
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₅₇H₆₄N₁₂O₉S	Melting Point	N/A
	MSDS	Chinese USA	Flash Point	N/A

Use of G Protein Antagonist

G-Protein antagonist peptide is the substance P-related peptide that inhibits binding of G proteins to their receptors. G-Protein antagonist peptide competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.

Name	G-Protein antagonist peptide
Synonym	More Synonyms

Description	G-Protein antagonist peptide is the substance P-related peptide that inhibits binding of G proteins to their receptors. G-Protein antagonist peptide competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.
Related Catalog	Signaling Pathways >> Neuronal Signaling >> mAChR Signaling Pathways >> GPCR/G Protein >> mAChR Signaling Pathways >> GPCR/G Protein >> Adrenergic Receptor

Molecular Formula	C₅₇H₆₄N₁₂O₉S
Molecular Weight	1093.26000
Exact Mass	1092.46000
PSA	362.55000
LogP	6.16720

Personal Protective Equipment	Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter
Safety Phrases	22-24/25
RIDADR	NONH for all modes of transport
WGK Germany	3

G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding.

J. Biol. Chem. 267 , 16237, (1992)

A substance P (SP) analog, [D-Pro4,D-Trp7,9,10] SP4-11, is known to inhibit the actions of various structurally unrelated messenger molecules as well as SP. Our studies on the effects of this peptide ...

PYR-GLN-D-TRP-PHE-D-TRP-D-TRP-MET-NH2

pglu-gln-d-trp-phe-d-trp-d-trp-met-nh2

G PROTEIN ANTAGONIST

PROTEIN G ANTAGONIST 2

GP ANTAGONIST-2

pGlu-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH2

[pGlu5,D-Trp7,9,10]-Substance P Fragment 5-11

G-PROTEIN ANTAGONIST-2