4,4,4-三氟-1-(2-呋喃基)-1,3-丁二酮
4,4,4-三氟-1-(2-呋喃基)-1,3-丁二酮结构式
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常用名 | 4,4,4-三氟-1-(2-呋喃基)-1,3-丁二酮 | 英文名 | Perfluoroacetyl(2-furoyl)methane |
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| CAS号 | 326-90-9 | 分子量 | 206.119 | |
| 密度 | 1.4±0.1 g/cm3 | 沸点 | 229.7±35.0 °C at 760 mmHg | |
| 分子式 | C8H5F3O3 | 熔点 | 19-21ºC(lit.) | |
| MSDS | 中文版 美版 | 闪点 | 92.7±25.9 °C |
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Bioorg. Med. Chem. Lett. 20 , 2622-4, (2010) 4,7-Dichloro-1-benzothien-2-yl sulfonylaminomethyl boronic acid (DSABA, Compound I) was discovered as the first boronic acid-based class D beta-lactamase inhibitor. It exhibited an IC(50) of 5.6 microM against OXA-40. The compound also inhibited class A and C... |
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