CPI-4203
Modify Date: 2024-01-11 01:07:47
CPI-4203 structure
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Common Name | CPI-4203 | ||
|---|---|---|---|---|
| CAS Number | 1628214-07-2 | Molecular Weight | 278.309 | |
| Density | 1.3±0.1 g/cm3 | Boiling Point | 499.4±55.0 °C at 760 mmHg | |
| Molecular Formula | C16H14N4O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 255.8±31.5 °C | |
Use of CPI-4203CPI-4203 is a potent KDM5A inhibitor with an IC50 of 250 nM. CPI-4203 is competitive with 2-oxoglutarate (2-OG). CPI-4203 is structurally related to CPI-455 (HY-100421) but is less potent[1]. |
| Name | 6-Ethyl-5-(2-methylphenyl)-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carbonitrile |
|---|---|
| Synonym | More Synonyms |
| Description | CPI-4203 is a potent KDM5A inhibitor with an IC50 of 250 nM. CPI-4203 is competitive with 2-oxoglutarate (2-OG). CPI-4203 is structurally related to CPI-455 (HY-100421) but is less potent[1]. |
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| Related Catalog | |
| Target |
IC50: 250 nM (KDM5A)[1] |
| References |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 499.4±55.0 °C at 760 mmHg |
| Molecular Formula | C16H14N4O |
| Molecular Weight | 278.309 |
| Flash Point | 255.8±31.5 °C |
| Exact Mass | 278.116760 |
| LogP | 2.58 |
| Vapour Pressure | 0.0±1.3 mmHg at 25°C |
| Index of Refraction | 1.670 |
| 6-Ethyl-5-(2-methylphenyl)-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carbonitrile |
| Pyrazolo[1,5-a]pyrimidine-3-carbonitrile, 6-ethyl-4,7-dihydro-5-(2-methylphenyl)-7-oxo- |