TUG-1375
Modify Date: 2024-01-10 22:54:41
TUG-1375 structure
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Common Name | TUG-1375 | ||
|---|---|---|---|---|
| CAS Number | 2247372-59-2 | Molecular Weight | 442.92 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C22H19ClN2O4S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of TUG-1375TUG-1375 is an agonist of free fatty acid receptor 2 (FFA2/GPR43), with a pKi of 6.69. TUG-1375 is inactive on FFA3, FFA4, PPARα, PPARγ, PPARδ, LXRα or LXRβ[1]. |
| Name | TUG-1375 |
|---|
| Description | TUG-1375 is an agonist of free fatty acid receptor 2 (FFA2/GPR43), with a pKi of 6.69. TUG-1375 is inactive on FFA3, FFA4, PPARα, PPARγ, PPARδ, LXRα or LXRβ[1]. |
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| Related Catalog | |
| Target |
pKi: 6.69 (FFA2)[1] |
| In Vitro | TUG-1375 exhibits pEC50 of 7.11 in the cAMP FFA2 assay, also active on murine FFA2 orthologue (pEC50, 6.44 ± 0.13 in the cAMP assay)[1]. |
| References |
| Molecular Formula | C22H19ClN2O4S |
|---|---|
| Molecular Weight | 442.92 |
| Storage condition | 2-8℃ |