PKCiota-IN-2

Modify Date: 2025-08-27 14:01:43

PKCiota-IN-2 Structure
PKCiota-IN-2 structure
Common Name PKCiota-IN-2
CAS Number 2230055-52-2 Molecular Weight 395.46
Density N/A Boiling Point N/A
Molecular Formula C24H21N5O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of PKCiota-IN-2


PKCiota-IN-2 is a potent PKCiota (PKC-ι) inhibitor with an IC50 of 2.8 nM. PKCiota-IN-2 also inhibits PKC-α and PKC-ε with IC50s of 71 nM and 350 nM, respectively[1].

 Names

Name PKCiota-IN-2

 PKCiota-IN-2 Biological Activity

Description PKCiota-IN-2 is a potent PKCiota (PKC-ι) inhibitor with an IC50 of 2.8 nM. PKCiota-IN-2 also inhibits PKC-α and PKC-ε with IC50s of 71 nM and 350 nM, respectively[1].
Related Catalog
Target

PKCι:2.8 nM (IC50)

PKCα:71 nM (IC50)

PKCε:350 nM (IC50)

References

[1]. Jacek Kwiatkowski, et al. Fragment-Based Drug Discovery of Potent Protein Kinase C Iota Inhibitors. J Med Chem. 2018 May 24;61(10):4386-4396.

 Chemical & Physical Properties

Molecular Formula C24H21N5O
Molecular Weight 395.46
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.
Top Suppliers:I want be here



Get all suppliers and price by the below link:

PKCiota-IN-2 suppliers

PKCiota-IN-2 price