CBP-IN-1

Modify Date: 2025-10-01 01:29:51

CBP-IN-1 Structure
CBP-IN-1 structure
Common Name CBP-IN-1
CAS Number 1936431-44-5 Molecular Weight 509.59
Density N/A Boiling Point N/A
Molecular Formula C27H33F2N7O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CBP-IN-1


CBP-IN-1 (compound 12) is a potent CBP inhibitor, with an IC50 of 1.5 nM. CBP-IN-1 also inhibits CBP BRET and BRD4(1), with IC50 values of 690 and 3100 nM, respectively[1].

 Names

Name CBP-IN-1

 CBP-IN-1 Biological Activity

Description CBP-IN-1 (compound 12) is a potent CBP inhibitor, with an IC50 of 1.5 nM. CBP-IN-1 also inhibits CBP BRET and BRD4(1), with IC50 values of 690 and 3100 nM, respectively[1].
Related Catalog
References

[1]. Romero FA, et al. GNE-781, A Highly Advanced Potent and Selective Bromodomain Inhibitor of Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP). J Med Chem. 2017 Nov 22;60(22):9162-9183.  

 Chemical & Physical Properties

Molecular Formula C27H33F2N7O
Molecular Weight 509.59
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.
Top Suppliers:I want be here