ATR-IN-13

Names

[ CAS No. ]:
2758113-84-5

[ Name ]:
ATR-IN-13

Biological Activity

[Description]:

ATR-IN-13 (compound A9) is a potent ATR kinase inhibitor, with an IC50 of 2 nM. ATR-IN-13 can be used for ATR kinase mediated diseases research, such as proliferative diseases and cancer[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Cell Cycle/DNA Damage >> ATM/ATR
Signaling Pathways >> PI3K/Akt/mTOR >> ATM/ATR

[Target]

ATR:2 nM (IC50)


[References]

[1]. Xiangling Zheng, et al. Pyrazolopyrimidine compounds as ATR kinase inhibitors. CN113929688A.

Chemical & Physical Properties

[ Molecular Formula ]:
C24H24FN9O

[ Molecular Weight ]:
473.51


Related Compounds