AHR antagonist 4

Modify Date: 2024-01-15 19:07:46

AHR antagonist 4 Structure
AHR antagonist 4 structure
Common Name AHR antagonist 4
CAS Number 2242465-58-1 Molecular Weight 488.34
Density N/A Boiling Point N/A
Molecular Formula C20H14F6N4O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of AHR antagonist 4


AHR antagonist 4 is a 2-heteroaryl-3-oxo-2,3-dihydropyridazine-4-carboxamide compound and a potent aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1, example 293, has an IC50 of 82.2 nM. AHR antagonist 4 has anti-cancer effects[1].

 Names

Name AHR antagonist 4

 AHR antagonist 4 Biological Activity

Description AHR antagonist 4 is a 2-heteroaryl-3-oxo-2,3-dihydropyridazine-4-carboxamide compound and a potent aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1, example 293, has an IC50 of 82.2 nM. AHR antagonist 4 has anti-cancer effects[1].
Related Catalog
Target

IC50: 82.2 nM (Aryl hydrocarbon receptor (AHR))[1]

References

[1]. Ilona GUTCHER, et al. 2-heteroaryl-3-oxo-2,3-dihydropyridazine-4-carboxamides for the treatment of cancer. WO2018146010A1.

 Chemical & Physical Properties

Molecular Formula C20H14F6N4O4
Molecular Weight 488.34