Journal of Peptide Science 2015-05-01

Solid-phase synthesis of C-terminal azapeptides.

Ngoc-Duc Doan, Jinqiang Zhang, Mariam Traoré, Winnie Kamdem, William D Lubell

Index: J. Pept. Sci. 21 , 387-91, (2015)

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Abstract

The solid-phase synthesis of azapeptides possessing a C-terminal aza-residue has been accomplished by a protocol featuring regioselective alkylation of benzhydrylidene-aza-glycinamide and illustrated by the syntheses of [aza-Lys(6)] growth-hormone-releasing peptide-6 analogs.Copyright © 2015 European Peptide Society and John Wiley & Sons, Ltd.