dynorphin (1-11), Pro(10)-
Modify Date: 2024-02-07 00:29:09
dynorphin (1-11), Pro(10)- structure
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Common Name | dynorphin (1-11), Pro(10)- | ||
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| CAS Number | 94596-26-6 | Molecular Weight | 1362.62000 | |
| Density | 1.42±0.1 g/cm3 (20 °C, 760 mmHg) | Boiling Point | N/A | |
| Molecular Formula | C63H103N21O13 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of dynorphin (1-11), Pro(10)-[DPro10] Dynorphin A (1-11), porcine, a N-Alkylated derivative, is a potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine has analgesic property[1][2]. |
| Name | α-Neoendorphin (swine), 7-L-arginine-8-L-isoleucine-8a-endo-L-arginine-9-D-proline |
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| Synonym | More Synonyms |
| Description | [DPro10] Dynorphin A (1-11), porcine, a N-Alkylated derivative, is a potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine has analgesic property[1][2]. |
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| Related Catalog | |
| In Vitro | [DPro10] Dynorphin A (1-11), porcine has inhibition of adenylyl cyclase activity in k-opioid receptor-expressing CHO cells with an IC50 value of 0.12 nM[1]. |
| In Vivo | [DPro10] Dynorphin A (1-11), porcine (ICV) has analgesic effects involving thermal cutaneous (tail-flick) and chemical visceral (AcOH-induced writhing) stimuli, in which mu and kappa receptors are known to be activated differentially[2]. |
| Density | 1.42±0.1 g/cm3 (20 °C, 760 mmHg) |
|---|---|
| Molecular Formula | C63H103N21O13 |
| Molecular Weight | 1362.62000 |
| Exact Mass | 1361.80000 |
| PSA | 577.48000 |
| LogP | 4.64670 |
| DYNORPHIN (1-11),PRO(10)- |
| YGGFLRRIRDPK |
| α-Neoendorphin (pig), 7-L-arginine-8-L-isoleucine-8a-endo-L-arginine-9-D-proline- |