Adenosine receptor inhibitor 2

Modify Date: 2025-09-01 17:04:47

Adenosine receptor inhibitor 2 Structure
Adenosine receptor inhibitor 2 structure
 Common Name Adenosine receptor inhibitor 2
CAS Number 2550401-76-6 Molecular Weight 406.28
Density N/A Boiling Point N/A
Molecular Formula C17H20BrN5O2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Adenosine receptor inhibitor 2


Adenosine receptor inhibitor 2 (compound 14b) is a potent AR (adenosine receptor) inhibitor. Adenosine receptor inhibitor 2 shows dual affinity toward A1/A2A ARs with higher affinity for the A1- than the A2AAR. Adenosine receptor inhibitor 2 has Ki values of 52.2 nM for the A1AR and 167 nM for the A2AAR[1].

 Names

Name Adenosine receptor inhibitor 2

 Adenosine receptor inhibitor 2 Biological Activity

Description Adenosine receptor inhibitor 2 (compound 14b) is a potent AR (adenosine receptor) inhibitor. Adenosine receptor inhibitor 2 shows dual affinity toward A1/A2A ARs with higher affinity for the A1- than the A2AAR. Adenosine receptor inhibitor 2 has Ki values of 52.2 nM for the A1AR and 167 nM for the A2AAR[1].
Related Catalog
Target

A1AR:52.2 ± 8.5 nM (Ki)

A2AR:167 ± 22 nM (Ki)

hA2B:>1000 nM (Ki)

Adenosine A3 receptor:>1000 nM (Ki)

References

[1]. Załuski M, et al. 8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation. Bioorg Chem. 2020 Aug;101:104033.

 Chemical & Physical Properties

Molecular Formula C17H20BrN5O2
Molecular Weight 406.28
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Chemsrc provides Adenosine receptor inhibitor 2(CAS#:2550401-76-6) MSDS, density, melting point, boiling point, structure, formula, molecular weight etc. Articles of Adenosine receptor inhibitor 2 are included as well.>> amp version: Adenosine receptor inhibitor 2

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