Adenosine receptor antagonist 1

Modify Date: 2024-01-11 19:31:05

Adenosine receptor antagonist 1 Structure
Adenosine receptor antagonist 1 structure
Common Name Adenosine receptor antagonist 1
CAS Number 2682930-40-9 Molecular Weight 447.85
Density N/A Boiling Point N/A
Molecular Formula C22H15ClFN7O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Adenosine receptor antagonist 1


Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aRthan A2bR.

 Names

Name Adenosine receptor antagonist 1

 Adenosine receptor antagonist 1 Biological Activity

Description Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aRthan A2bR.
Related Catalog
Target

A2AR:0.29 nM (IC50)

References

[1]. Lamb ML, et al. Triazole compounds as adenosine receptor antagonists. WO2021156439A1.

 Chemical & Physical Properties

Molecular Formula C22H15ClFN7O
Molecular Weight 447.85