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Adenosine receptor antagonist 1

Names

[ CAS No. ]:
2682930-40-9

[ Name ]:
Adenosine receptor antagonist 1

Biological Activity

[Description]:

Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aRthan A2bR.

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> GPCR/G Protein >> Adenosine Receptor

[Target]

A2AR:0.29 nM (IC50)


[References]

[1]. Lamb ML, et al. Triazole compounds as adenosine receptor antagonists. WO2021156439A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C22H15ClFN7O

[ Molecular Weight ]:
447.85

Related Compounds