CSNK1-IN-1 structure
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Common Name | CSNK1-IN-1 | ||
|---|---|---|---|---|
| CAS Number | 2468784-55-4 | Molecular Weight | 533.54 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C29H26F3N5O2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of CSNK1-IN-1CSNK1-IN-1 is a CSNK1A1 inhibitor. CSNK1-IN-1 has inhibitory activity for CSNK1A1 kinase with IC50 values of 21 μM. CSNK1-IN-1 can be used for the research of proliferative disorders[1]. |
| Name | CSNK1-IN-1 |
|---|
| Description | CSNK1-IN-1 is a CSNK1A1 inhibitor. CSNK1-IN-1 has inhibitory activity for CSNK1A1 kinase with IC50 values of 21 μM. CSNK1-IN-1 can be used for the research of proliferative disorders[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 21 μM (CSNK1A1 kinase)[1] |
| In Vitro | CSNK1-IN-1 对 CSNK1A1, CSNK1D 和 CSNK1A1 (高 ATP) 具有抑制活性,IC50 值分别为 21 μM, 29.7 μM 和 1.5 nM[1]。< br / >CSNK1-IN-1 对野生型 EGFR 激酶表现出低抑制作用,其 IC50 值为 >20 nM[1]。 |
| References |
| Molecular Formula | C29H26F3N5O2 |
|---|---|
| Molecular Weight | 533.54 |
| InChIKey | IKATWWUGCJFQJV-OAQYLSRUSA-N |
| SMILES | CN1CCc2[nH]c(-c3ccnc(NC(=O)C(CC(F)F)c4ccc(F)cc4)c3)c(Nc3ccccc3)c2C1=O |