FFA1 agonist-1

Modify Date: 2024-01-04 20:14:38

FFA1 agonist-1 Structure
FFA1 agonist-1 structure
Common Name FFA1 agonist-1
CAS Number 2417231-16-2 Molecular Weight 458.03
Density N/A Boiling Point N/A
Molecular Formula C27H36ClNO3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of FFA1 agonist-1


FFA1 agonist-1 (Compound 17a) is an orally active fatty acid receptor 1 (FFA1) agonist with an EC50 of 0.75 μM. FFA1 agonist-1 can be used for type 2 diabetes mellitus research[1].

 Names

Name FFA1 agonist-1

 FFA1 agonist-1 Biological Activity

Description FFA1 agonist-1 (Compound 17a) is an orally active fatty acid receptor 1 (FFA1) agonist with an EC50 of 0.75 μM. FFA1 agonist-1 can be used for type 2 diabetes mellitus research[1].
Related Catalog
Target

EC50: 0.75 μM (FFA1)[1]

In Vivo FFA1 agonist-1 (Compound 17a) (0-25 mg/kg; p.o.) reduces the plasma glucose levels in a dose-dependent manner in mice[1].
References

[1]. Kuranov SO, et al. Exploring bulky natural and natural-like periphery in the design of p-(benzyloxy)phenylpropionic acid agonists of free fatty acid receptor 1 (GPR40). Bioorg Chem. 2020 Jun;99:103830.

 Chemical & Physical Properties

Molecular Formula C27H36ClNO3
Molecular Weight 458.03