AT-090 structure
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Common Name | AT-090 | ||
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CAS Number | 2099681-59-9 | Molecular Weight | 354.494 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C22H30N2O2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of AT-090AT-090 is a novel potent, selective nociceptin/orphanin FQ receptor (NOP receptor) agonist with Ki of 5.61 nM; displays >15-fold selectivity over mu, and >40-fold over kappa opioid receptors; induces concentration dependent contractions of the mouse colon tissues with potency and efficacy similar to N/OFQ; a useful pharmacological tool for investigating the therapeutic potential of NOP partial agonists. |
Name | AT-090 |
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Description | AT-090 is a novel potent, selective nociceptin/orphanin FQ receptor (NOP receptor) agonist with Ki of 5.61 nM; displays >15-fold selectivity over mu, and >40-fold over kappa opioid receptors; induces concentration dependent contractions of the mouse colon tissues with potency and efficacy similar to N/OFQ; a useful pharmacological tool for investigating the therapeutic potential of NOP partial agonists. |
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References | References 1. Ferrari F, et al. Eur J Pharmacol. 2016 Dec 15;793:1-13. 2. Asth L, et al. Neuropharmacology. 2016 Jun;105:434-442. View Related Products by Target Opioid Receptor |
Molecular Formula | C22H30N2O2 |
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Molecular Weight | 354.494 |