ZEN-3219 structure
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Common Name | ZEN-3219 | ||
|---|---|---|---|---|
| CAS Number | 1952264-34-4 | Molecular Weight | 322.36 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C19H18N2O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of ZEN-3219ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4[1]. |
| Name | ZEN-3219 |
|---|
| Description | ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4[1]. |
|---|---|
| Related Catalog | |
| Target |
BRD4 (BD1):0.48 μM (IC50) BRD4 (BD2):0.16 μM (IC50) BRD4(BD1BD2):0.47 μM (IC50) |
| References |
| Molecular Formula | C19H18N2O3 |
|---|---|
| Molecular Weight | 322.36 |
| InChIKey | IELJHNIVCXDKQD-UHFFFAOYSA-N |
| SMILES | Cc1noc(C)c1-c1ccc(=O)n(Cc2ccc(C3CO3)cc2)c1 |
| Hazard Codes | Xi |
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