Name | ZEN-3411 |
---|
Description | ZEN-3411 is a BET inhibitor with IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3411 can be used to form PROTACs to induce degradation of BRD4[1]. |
---|---|
Related Catalog | |
Target |
BRD4 (BD1):0.05 μM (IC50) BRD4 (BD2):0.05 μM (IC50) BRD4(BD1BD2):0.06 μM (IC50) |
References |
Molecular Formula | C21H20N4O2 |
---|---|
Molecular Weight | 360.41 |
Hazard Codes | Xi |
---|