PI3Kα inhibitor 1
Modify Date: 2025-08-22 22:40:00
PI3Kα inhibitor 1 structure
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Common Name | PI3Kα inhibitor 1 | ||
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| CAS Number | 1235449-52-1 | Molecular Weight | 507.568 | |
| Density | 1.5±0.1 g/cm3 | Boiling Point | N/A | |
| Molecular Formula | C23H25N9O3S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PI3Kα inhibitor 1PI3Kα inhibitor 1 is a selective PI3Kα inhibitor extracted from patent US/20120088764A1, Compound 243, has an IC50<0.1 μM, PI3Kα inhibitor 1 also inhibits HDAC (0.1 μM≤IC50≤1 μM) . |
| Name | N-Hydroxy-2-[methyl({2-[6-(methylamino)-3-pyridinyl]-4-(4-morpholinyl)thieno[3,2-d]pyrimidin-6-yl}methyl)amino]-5-pyrimidinecarboxamide |
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| Synonym | More Synonyms |
| Description | PI3Kα inhibitor 1 is a selective PI3Kα inhibitor extracted from patent US/20120088764A1, Compound 243, has an IC50<0.1 μM, PI3Kα inhibitor 1 also inhibits HDAC (0.1 μM≤IC50≤1 μM) . |
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| Related Catalog | |
| Target |
PI3Kα:0.1 μM (IC50) HDAC:0.1 μM (IC50) |
| References |
| Density | 1.5±0.1 g/cm3 |
|---|---|
| Molecular Formula | C23H25N9O3S |
| Molecular Weight | 507.568 |
| Exact Mass | 507.180115 |
| LogP | 2.31 |
| Index of Refraction | 1.728 |
| N-Hydroxy-2-[methyl({2-[6-(methylamino)-3-pyridinyl]-4-(4-morpholinyl)thieno[3,2-d]pyrimidin-6-yl}methyl)amino]-5-pyrimidinecarboxamide |
| 5-Pyrimidinecarboxamide, N-hydroxy-2-[methyl[[2-[6-(methylamino)-3-pyridinyl]-4-(4-morpholinyl)thieno[3,2-d]pyrimidin-6-yl]methyl]amino]- |
| CUDC-908 |
| PI3Kα inhibitor 1 |
| BEBT-908 |