Pim1/AKK1-IN-1
Modify Date: 2024-01-05 17:34:06
Pim1/AKK1-IN-1 structure
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Common Name | Pim1/AKK1-IN-1 | ||
|---|---|---|---|---|
| CAS Number | 1093222-27-5 | Molecular Weight | 339.35000 | |
| Density | 1.42 | Boiling Point | N/A | |
| Molecular Formula | C20H13N5O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Pim1/AKK1-IN-1Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK. |
| Name | N-[5-(4-cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide |
|---|---|
| Synonym | More Synonyms |
| Description | Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK. |
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| Related Catalog | |
| Target |
Kd: 35 nM (Pim1), 53 nM (AKK1), 75 nM (MST2), 380 nM (LKB1) |
| In Vitro | Pim1/AKK1-IN-1 is multi-kinase inhibitor, and has Kd of 380 nM against LKB1 and 53 nM against AAK1[1]. |
| References |
| Density | 1.42 |
|---|---|
| Molecular Formula | C20H13N5O |
| Molecular Weight | 339.35000 |
| Exact Mass | 339.11200 |
| PSA | 97.95000 |
| LogP | 4.13288 |
| Storage condition | 2-8℃ |
| 3-Pyridinecarboxamide,N-[5-(4-cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl] |
| CS-0342 |
| LKB1 (AAK1 dual inhibitor) |
| N-[5-(4-Cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-3-pyridinecarboxamide |
| LKB1(AAK1 dual inhibitor)||3-Pyridinecarboxamide,N-[5-(4-cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl] |
| Pim1/AKK1-IN-1 |