502486-89-7
502486-89-7 structure
- Name: NIDA-41020
- Chemical Name: 1-(2,4-dichlorophenyl)-5-(4-methoxyphenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
- CAS Number: 502486-89-7
- Molecular Formula: C23H24Cl2N4O2
- Molecular Weight: 459.36800
- Catalog: Signaling Pathways GPCR/G Protein Cannabinoid Receptor
- Create Date: 2016-02-17 02:44:00
- Modify Date: 2025-08-25 16:58:17
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NIDA-41020 is a potent and selective cannabinoid receptor 1(CB1) antagonist with a Ki of 4.1 nM. NIDA-41020 was designed as a potential radioligand for use in positron emission tomography (PET)[1].
| Name | 1-(2,4-dichlorophenyl)-5-(4-methoxyphenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide |
|---|---|
| Synonyms |
1-(2,4-Dichlorophenyl)-5-(4-methoxyphenyl)-4-methyl-N-(1-piperidinyl)-1H-pyrazole-3-carboxamide
Roxindole hydrochloride |
| Description | NIDA-41020 is a potent and selective cannabinoid receptor 1(CB1) antagonist with a Ki of 4.1 nM. NIDA-41020 was designed as a potential radioligand for use in positron emission tomography (PET)[1]. |
|---|---|
| Related Catalog | |
| Target |
CB1:4.1 nM (Ki) |
| References |
| Molecular Formula | C23H24Cl2N4O2 |
|---|---|
| Molecular Weight | 459.36800 |
| Exact Mass | 458.12800 |
| PSA | 59.39000 |
| LogP | 5.62260 |
| Storage condition | 2-8°C |
| Symbol |
GHS06 |
|---|---|
| Signal Word | Danger |
| Hazard Statements | H300-H315-H319-H335 |
| Precautionary Statements | P261-P264-P301 + P310-P305 + P351 + P338 |
| Personal Protective Equipment | Eyeshields;Faceshields;Gloves;type P2 (EN 143) respirator cartridges |
| Risk Phrases | 25-36/37/38 |
| Safety Phrases | 26-45 |
| RIDADR | UN 2811 6.1 / PGIII |