| Name | PKN1/2-IN-1 |
|---|
| Description | PKN1/2-IN-1 is a potent, cell penetrant and selective PKN2 (PRK2) inhibitor (IC50=16 nM; Ki=8 nM)[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 16 nM, Ki: 8 nM (PKN2)[1] IC50: 108 nM, Ki: 210 nM (PKN1)[1]. |
| References |
| Molecular Formula | C14H15N3O |
|---|---|
| Molecular Weight | 241.29 |