DRAK2-IN-16

Names

[ Name ]:
DRAK2-IN-16

Biological Activity

[Description]:

DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively.DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM)[1].

[Related Catalog]:

Research Areas >> Others

Signaling Pathways >> Apoptosis >> DAPK

[Target]

IC50: 3 nM (DRAK2); 51 nM (DRAK1); 1.8 μM (DRPK2); 2.3 μM (DRAK2); 1.8 μM (DRPK3)[1]

[References]

[1]. Aranda-González I, et al. Evaluation of the Antihyperglycemic Effect of Minor Steviol Glycosides in Normoglycemic and Induced-Diabetic Wistar Rats. J Med Food. 2016 Sep;19(9):844-52.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₁H₂₀N₄O₃

[ Molecular Weight ]:
376.41

Safety Information

[ Hazard Codes ]:
Xi

Related Compounds

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