| Name | DRAK2-IN-1 |
|---|
| Description | DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively.DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM)[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 3 nM (DRAK2); 51 nM (DRAK1); 1.8 μM (DRPK2); 2.3 μM (DRAK2); 1.8 μM (DRPK3)[1] |
| References |
| Molecular Formula | C21H20N4O3 |
|---|---|
| Molecular Weight | 376.41 |
| Hazard Codes | Xi |
|---|